SCHEMBL4639398

SCHEMBL4639398

CC(C)(C)[Si](C)(C)OCc1onc(-c2c(Cl)cccc2Cl)c1C(=O)c1nnn(Cc2cc(C(F)(F)F)cc(C(F)(F)F)c2)c1N1CCOCC1

nearest known ligand 0.37

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 3/20 0.37
KDM4E B2RXH2 1/20 0.36
ALDH1A1 P00352 4/20 0.36
TSHR P16473 2/20 0.36
NPSR1 Q6W5P4 1/20 0.34
NR1H4 Q96RI1 1/20 0.34
PPARD Q03181 1/20 0.34
TACR1 P25103 2/20 0.33
L3MBTL1 Q9Y468 2/20 0.33
TP53 P04637 1/20 0.33
MAPT P10636 1/20 0.33
MEN1 O00255 1/20 0.32
POLB P06746 1/20 0.32
KCNH2 Q12809 2/20 0.32
TDP1 Q9NUW8 1/20 0.32
SLC16A3 O15427 1/20 0.32
SLC16A1 P53985 1/20 0.32
MCTS1 Q9ULC4 1/20 0.32
DHODH Q02127 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4638841 0.93 TACR1 (0.34) KMT2AKDM4EALDH1A1TSHRTACR1
SCHEMBL4639495 0.89 TACR1 (0.31) KMT2AALDH1A1TSHRTACR1L3MBTL1
SCHEMBL4638040 0.88 ALDH1A1 (0.31) ALDH1A1TACR1L3MBTL1TDP1
SCHEMBL4638555 0.88 CNR1 (0.32) ALDH1A1L3MBTL1TDP1
SCHEMBL4637966 0.88 KMT2A (0.41) KMT2AALDH1A1NR1H4PPARDTACR1
SCHEMBL4638545 0.86 ALDH1A1 (0.38) KMT2AKDM4EALDH1A1TSHRTACR1
SCHEMBL4639400 0.84 NR1H4 (0.37) KMT2AKDM4EALDH1A1TSHRNPSR1
SCHEMBL4637842 0.82 TACR1 (0.36) KMT2AKDM4EALDH1A1TSHRTACR1
SCHEMBL4637694 0.81 EPAS1 (0.39) KMT2AKDM4EALDH1A1TSHRTACR1
SCHEMBL4637876 0.81 EPAS1 (0.39) KMT2AKDM4EALDH1A1TSHRTACR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1501808-B1 TACHYKININ RECEPTOR ANTAGONISTS LILLY CO ELI (US) 2008-07-02 EP disclosed