SCHEMBL4640260

SCHEMBL4640260

O=C(O)CC(NC(=O)OCc1ccccc1)n1cnc2c(N3CCC(C(=O)NC4=NCCCN4)CC3)ncnc21

nearest known ligand 0.43

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
ITGB3 P05106 11/20 0.43
ITGAV P06756 11/20 0.43
ITGA2B P08514 3/20 0.43
MAPT P10636 1/20 0.38
KMT2A Q03164 2/20 0.38
MEN1 O00255 1/20 0.38
CNR1 P21554 1/20 0.38
CNR2 P34972 1/20 0.38
UBE2N P61088 1/20 0.37
ITGB5 P18084 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6810562 0.92 ITGB3 (0.41) ITGB3ITGAVITGA2BMAPTKMT2A
SCHEMBL6805470 0.88 TDP1 (0.36) ITGB3ITGAVITGA2BMAPTKMT2A
SCHEMBL6803682 0.86 ITGB3 (0.45) ITGB3ITGAVITGA2BMAPTKMT2A
SCHEMBL4640251 0.86 ITGB3 (0.49) ITGB3ITGAVITGA2BITGB5
SCHEMBL6802245 0.85 ITGB3 (0.49) ITGB3ITGAVITGA2BITGB5
SCHEMBL6811105 0.85 CNR1 (0.44) ITGB3ITGAVCNR1CNR2
SCHEMBL7702988 0.82 ITGB3 (0.44) ITGB3ITGAVITGA2BMAPTITGB5
SCHEMBL4644035 0.82 ITGB3 (0.44) ITGB3ITGAVITGA2BMAPTITGB5
SCHEMBL6806629 0.82 TDP1 (0.35) ITGB3ITGAVITGA2BMAPTKMT2A
SCHEMBL6804912 0.82 ITGB3 (0.45) ITGB3ITGAVCNR1CNR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0853084-B1 Substituted purine derivatives as vitronectin receptor antagonists HOECHST AG (DE) 2008-08-13 EP claimed
US-6723727-B1 VITRONECTIN RECEPTOR ANTAGONISTS; INHIBITORS OF BONE RESORPTION; OSTEOPOROSIS HOECHST AKTIENGESELLSCHAFT (DE) 2004-04-20 US claimed
US-6723727-B1 VITRONECTIN RECEPTOR ANTAGONISTS; INHIBITORS OF BONE RESORPTION; OSTEOPOROSIS HOECHST AKTIENGESELLSCHAFT (DE) 2004-04-20 US disclosed