SCHEMBL4640795

SCHEMBL4640795

CC(C)(C)OC(=O)[C@H](Cn1cnc2c(Sc3cccc(N)c3)ncnc21)NC(=O)OCc1ccccc1

nearest known ligand 0.38

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
SLC29A1 Q99808 1/20 0.38
SYK P43405 1/20 0.36
JAK2 O60674 1/20 0.35
ADORA3 P0DMS8 1/20 0.35
ADORA2A P29274 1/20 0.35
ADORA2B P29275 1/20 0.35
ADORA1 P30542 1/20 0.35
ITGB3 P05106 1/20 0.34
ITGAV P06756 1/20 0.34
CTSK P43235 3/20 0.34
CTSL P07711 1/20 0.34
CTSB P07858 1/20 0.34
CTSS P25774 1/20 0.34
DOT1L Q8TEK3 1/20 0.34
ALDH1A1 P00352 1/20 0.34
CYP1A2 P05177 1/20 0.34
MMP13 P45452 2/20 0.34
MAPT P10636 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6807080 0.91 ITGB3 (0.40) ITGB3ITGAVDOT1LALDH1A1CYP1A2
SCHEMBL4641533 0.87 ITGB3 (0.42) SLC29A1SYKJAK2ITGB3ITGAV
SCHEMBL6807305 0.83 SYK (0.36) SLC29A1SYKJAK2ADORA3ADORA2A
SCHEMBL6016459 0.81 HDAC6 (0.43) SYKITGB3ITGAVCTSKCTSL
SCHEMBL6016455 0.81 HDAC6 (0.43) SYKITGB3ITGAVCTSKCTSL
SCHEMBL6807303 0.80 JAK2 (0.36) SLC29A1SYKJAK2ALDH1A1
SCHEMBL6807083 0.79 CASP1 (0.37) DOT1L
SCHEMBL4640030 0.78 TDP1 (0.45) SYKADORA2AADORA1ITGB3ITGAV
SCHEMBL6807059 0.78 TDP1 (0.45) SYKADORA2AADORA1ITGB3ITGAV
SCHEMBL4641344 0.77 ITGB3 (0.48) ITGB3ITGAVMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0853084-B1 Substituted purine derivatives as vitronectin receptor antagonists HOECHST AG (DE) 2008-08-13 EP disclosed
EP-0853084-A2 Substituted purine derivatives as vitronectin receptor antagonists HOECHST AKTIENGESELLSCHAFT (DE) 1998-07-15 EP disclosed