SCHEMBL4640844

SCHEMBL4640844

CC(C)(C)OC(=O)[C@H](Cn1cnc2c(N3CCC(CN)CC3)ncnc21)NC(=O)OCc1ccccc1

nearest known ligand 0.48

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
ITGB3 P05106 17/20 0.48
ITGAV P06756 17/20 0.48
ITGA2B P08514 1/20 0.43
ITGB5 P18084 1/20 0.43
ADORA3 P0DMS8 1/20 0.40
ADORA2A P29274 1/20 0.40
ADORA2B P29275 1/20 0.40
ADORA1 P30542 1/20 0.40
HRH4 Q9H3N8 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27524220 0.91 ITGB3 (0.46) ITGB3ITGAVITGA2BITGB5ADORA3
SCHEMBL4640164 0.91 ITGB3 (0.46) ITGB3ITGAVITGA2BITGB5ADORA3
SCHEMBL4641583 0.91 ITGB3 (0.55) ITGB3ITGAVITGA2BITGB5
SCHEMBL6810547 0.84 ITGB3 (0.40) ITGB3ITGAVADORA3ADORA2AADORA2B
SCHEMBL4644035 0.83 ITGB3 (0.44) ITGB3ITGAVITGA2BITGB5
SCHEMBL7702988 0.83 ITGB3 (0.44) ITGB3ITGAVITGA2BITGB5
SCHEMBL6016455 0.82 HDAC6 (0.43) ITGB3ITGAV
SCHEMBL6016459 0.82 HDAC6 (0.43) ITGB3ITGAV
SCHEMBL6811091 0.81 ITGB3 (0.53) ITGB3ITGAVITGA2BITGB5
SCHEMBL6016567 0.81 ITGAV (0.44) ITGB3ITGAVITGA2BITGB5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0853084-B1 Substituted purine derivatives as vitronectin receptor antagonists HOECHST AG (DE) 2008-08-13 EP disclosed
EP-0853084-A2 Substituted purine derivatives as vitronectin receptor antagonists HOECHST AKTIENGESELLSCHAFT (DE) 1998-07-15 EP disclosed