SCHEMBL4643663

SCHEMBL4643663

CN(C)CCN(C)c1nc2ccc(NC(=O)Oc3ccc(-c4ccc(F)cc4Cl)cc3)cc2s1

nearest known ligand 0.46

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.46
SMN1; SMN2 Q16637 2/20 0.46
HTT P42858 3/20 0.42
KMT2A Q03164 2/20 0.42
TMPRSS15 P98073 3/20 0.41
MCHR1 Q99705 1/20 0.40
LMNA P02545 2/20 0.39
MAPT P10636 4/20 0.39
HPGD P15428 1/20 0.39
HSD17B10 Q99714 1/20 0.39
AURKB Q96GD4 1/20 0.38
TP53 P04637 1/20 0.38
MEN1 O00255 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4643578 0.92 MCHR1 (0.44) ALDH1A1SMN1; SMN2HTTKMT2ATMPRSS15
SCHEMBL4641355 0.92 ALDH1A1 (0.44) ALDH1A1SMN1; SMN2HTTKMT2ATMPRSS15
SCHEMBL4644016 0.91 ALDH1A1 (0.43) ALDH1A1SMN1; SMN2HTTKMT2ATMPRSS15
SCHEMBL4641406 0.91 MAPT (0.42) ALDH1A1SMN1; SMN2HTTKMT2ATMPRSS15
SCHEMBL4641593 0.91 MAPT (0.46) ALDH1A1SMN1; SMN2KMT2ATMPRSS15MCHR1
SCHEMBL4647202 0.91 CACNA1B (0.44) ALDH1A1SMN1; SMN2KMT2ATMPRSS15MCHR1
SCHEMBL4641244 0.90 ALDH1A1 (0.45) ALDH1A1SMN1; SMN2HTTKMT2ATMPRSS15
SCHEMBL4641377 0.90 MCHR1 (0.45) TMPRSS15MCHR1
SCHEMBL4643026 0.89 MCHR1 (0.42) SMN1; SMN2KMT2ATMPRSS15MCHR1LMNA
SCHEMBL5244294 0.88 MCHR1 (0.47) ALDH1A1SMN1; SMN2HTTKMT2AMCHR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1828177-B1 NOVEL MCH RECEPTOR ANTAGONISTS LILLY CO ELI (US) 2008-08-13 EP claimed