SCHEMBL4647202

SCHEMBL4647202

CN(C)CCN(C)c1nc2ccc(NC(=O)Oc3ccc(-c4ccc(C(F)(F)F)cc4Cl)cc3)cc2s1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CACNA1B Q00975 2/20 0.44
CACNA1H O95180 1/20 0.44
MCHR1 Q99705 6/20 0.44
ADRA1D P25100 1/20 0.44
ADRA1A P35348 1/20 0.44
ADRA1B P35368 1/20 0.44
HTR2B P41595 1/20 0.44
AGPAT2 O15120 4/20 0.43
CSNK1D P48730 2/20 0.41
TMPRSS15 P98073 2/20 0.40
ALDH1A1 P00352 1/20 0.38
SMN1; SMN2 Q16637 1/20 0.38
MEN1 O00255 1/20 0.38
NPC1 O15118 1/20 0.38
USP2 O75604 1/20 0.38
LMNA P02545 1/20 0.38
TP53 P04637 1/20 0.38
CYP1A2 P05177 1/20 0.38
CYP3A4 P08684 1/20 0.38
CYP2D6 P10635 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4641377 0.92 MCHR1 (0.45) CACNA1BCACNA1HMCHR1ADRA1DADRA1A
SCHEMBL4643663 0.91 ALDH1A1 (0.46) MCHR1TMPRSS15ALDH1A1SMN1; SMN2MEN1
SCHEMBL4643578 0.90 MCHR1 (0.44) MCHR1TMPRSS15ALDH1A1SMN1; SMN2MEN1
SCHEMBL4641593 0.90 MAPT (0.46) MCHR1TMPRSS15ALDH1A1SMN1; SMN2MEN1
SCHEMBL4641406 0.90 MAPT (0.42) MCHR1TMPRSS15ALDH1A1SMN1; SMN2MEN1
SCHEMBL5246435 0.89 MCHR1 (0.54) CACNA1BCACNA1HMCHR1ADRA1DADRA1A
SCHEMBL4643026 0.88 MCHR1 (0.42) MCHR1TMPRSS15SMN1; SMN2MEN1LMNA
SCHEMBL4643038 0.85 MCHR1 (0.48) MCHR1TMPRSS15ALDH1A1SMN1; SMN2MEN1
SCHEMBL4645813 0.85 TMPRSS15 (0.41) MCHR1TMPRSS15ALDH1A1SMN1; SMN2MEN1
SCHEMBL4641355 0.84 ALDH1A1 (0.44) CACNA1BTMPRSS15ALDH1A1SMN1; SMN2MEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1828177-B1 NOVEL MCH RECEPTOR ANTAGONISTS LILLY CO ELI (US) 2008-08-13 EP claimed