SCHEMBL4644568

SCHEMBL4644568

CN1CCC(N(C)c2nc3cc(NC(=O)Oc4ccc(-c5ccc(Cl)cc5)s4)ccc3o2)CC1

nearest known ligand 0.39

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
CASP3 P42574 1/20 0.39
SENP8 Q96LD8 1/20 0.39
SENP7 Q9BQF6 1/20 0.39
SENP6 Q9GZR1 1/20 0.39
MCHR1 Q99705 3/20 0.38
MAPT P10636 3/20 0.38
KDR P35968 3/20 0.37
HDAC1 Q13547 1/20 0.37
HDAC2 Q92769 1/20 0.37
PTGS2 P35354 1/20 0.37
AGPAT2 O15120 2/20 0.36
TP53 P04637 2/20 0.36
RXFP1 Q9HBX9 1/20 0.36
PTGDR2 Q9Y5Y4 3/20 0.36
THRB P10828 1/20 0.36
FAAH O00519 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4646542 0.93 MCHR1 (0.41) MCHR1MAPTHDAC1HDAC2PTGS2
SCHEMBL4642981 0.93 NPC1 (0.38) MCHR1MAPTHDAC1HDAC2PTGS2
SCHEMBL4641252 0.92 PTGDR2 (0.39) MCHR1MAPTTP53PTGDR2THRB
SCHEMBL4643611 0.92 SMN1; SMN2 (0.39) MCHR1MAPTKDRAGPAT2TP53
SCHEMBL4641302 0.92 MAPT (0.42) MCHR1MAPTKDRPTGS2TP53
SCHEMBL4641260 0.91 MCHR1 (0.38) MCHR1KDRHDAC1HDAC2PTGDR2
SCHEMBL4641270 0.88 MAPT (0.40) MCHR1MAPTHDAC1HDAC2TP53
SCHEMBL4643502 0.84 PTGDR2 (0.40) MCHR1MAPTPTGDR2
SCHEMBL4641201 0.83 AGPAT2 (0.42) CASP3SENP8SENP7SENP6MAPT
SCHEMBL4641410 0.82 AGPAT2 (0.42) CASP3SENP8SENP7SENP6MCHR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1828177-B1 NOVEL MCH RECEPTOR ANTAGONISTS LILLY CO ELI (US) 2008-08-13 EP claimed