SCHEMBL46453

SCHEMBL46453

CCOC(=O)c1cc2nc(Cc3cccs3)[nH]c(=O)c2s1

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 3/20 0.50
SMN1; SMN2 Q16637 2/20 0.50
PDE5A O76074 1/20 0.49
CDC7 O00311 3/20 0.44
CCNE1 P24864 3/20 0.44
CDK2 P24941 3/20 0.44
ROCK1 Q13464 3/20 0.44
DBF4 Q9UBU7 3/20 0.44
TSHR P16473 3/20 0.43
LMNA P02545 1/20 0.43
ALDH1A1 P00352 1/20 0.41
PNP P00491 1/20 0.40
RXFP1 Q9HBX9 1/20 0.39
CTDSP1 Q9GZU7 1/20 0.39
TDP1 Q9NUW8 1/20 0.39
L3MBTL1 Q9Y468 1/20 0.39
HSD17B10 Q99714 2/20 0.39
NPC1 O15118 1/20 0.39
TP53 P04637 1/20 0.39
HPGD P15428 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL38373 0.85 PDE5A (0.61) KDM4ESMN1; SMN2PDE5ACDC7CCNE1
SCHEMBL38116 0.85 PDE5A (0.63) KDM4ESMN1; SMN2PDE5ATSHRLMNA
SCHEMBL4530199 0.84 SMN1; SMN2 (0.50) KDM4ESMN1; SMN2PDE5ATSHRLMNA
SCHEMBL46291 0.82 PDE5A (0.50) PDE5ACDC7CCNE1CDK2ROCK1
SCHEMBL10084040 0.81 PDE5A (0.59) KDM4ESMN1; SMN2PDE5ACDC7CCNE1
SCHEMBL46289 0.81 PDE5A (0.76) KDM4ESMN1; SMN2PDE5ACDC7CCNE1
SCHEMBL10083509 0.81 PDE5A (0.58) PDE5ACDC7CCNE1CDK2ROCK1
SCHEMBL38484 0.80 PDE5A (0.57) KDM4ESMN1; SMN2PDE5ACDC7CCNE1
SCHEMBL46296 0.77 PDE5A (0.56) KDM4ESMN1; SMN2PDE5ACDC7CCNE1
SCHEMBL4523121 0.76 KMT2A (0.64) KDM4ETSHRLMNAALDH1A1RXFP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012004900-A1 THIENOPYRIMIDINE COMPOUNDS ASKA PHARMACEUTICAL CO., LTD. (JP) 2012-01-12 WO disclosed