SCHEMBL4649044

SCHEMBL4649044

N#Cc1ccccc1Cc1cc2c(=O)c(C(=O)O)c[nH]c2cc1Cl

nearest known ligand 0.46

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
PRKAB2 O43741 6/20 0.46
PRKAG1 P54619 6/20 0.46
PRKAA2 P54646 6/20 0.46
PRKAA1 Q13131 6/20 0.46
PRKAG3 Q9UGI9 6/20 0.46
PRKAG2 Q9UGJ0 6/20 0.46
PRKAB1 Q9Y478 6/20 0.46
MDH2 P40926 2/20 0.45
ALDH1A1 P00352 1/20 0.45
HPGD P15428 1/20 0.45
SMN1; SMN2 Q16637 1/20 0.45
SNCA P37840 2/20 0.42
KDM4E B2RXH2 2/20 0.42
MEN1 O00255 1/20 0.41
ADRB2 P07550 1/20 0.41
RECQL P46063 1/20 0.41
KMT2A Q03164 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6713044 0.84 MDH2 (0.55) PRKAB2PRKAG1PRKAA2PRKAA1PRKAG3
SCHEMBL6717561 0.81 MDH2 (0.54) PRKAB2PRKAG1PRKAA2PRKAA1PRKAG3
SCHEMBL4650048 0.77 KDM4E (0.50) PRKAB2PRKAG1PRKAA2PRKAA1PRKAG3
SCHEMBL6714522 0.76 HTT (0.51) PRKAB2PRKAG1PRKAA2PRKAA1PRKAG3
SCHEMBL4649270 0.76 KDM4E (0.57) PRKAB2PRKAG1PRKAA2PRKAA1PRKAG3
SCHEMBL4649992 0.74 KDM4E (0.47) PRKAB2PRKAG1PRKAA2PRKAA1PRKAG3
SCHEMBL4650034 0.74 KDM4E (0.49) PRKAB2PRKAG1PRKAA2PRKAA1PRKAG3
SCHEMBL4650042 0.74 ALDH1A1 (0.58) PRKAB2PRKAG1PRKAA2PRKAA1PRKAG3
SCHEMBL4650661 0.73 ALDH1A1 (0.60) PRKAB2PRKAG1PRKAA2PRKAA1PRKAG3
SCHEMBL10955456 0.72 KDM4E (0.49) PRKAB2PRKAG1PRKAA2PRKAA1PRKAG3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1963271-A1 QUINOLONE M1 RECEPTOR POSITIVE ALLOSTERIC MODULATORS Merck & Co., Inc. (US) 2008-09-03 EP claimed
WO-2007067489-A1 QUINOLONE M1 RECEPTOR POSITIVE ALLOSTERIC MODULATORS MERCK & CO., INC. (US) 2007-06-14 WO claimed