SCHEMBL4649823

SCHEMBL4649823

O=C(O)c1c[nH]c(=O)c(Cc2ccccn2)c1

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 2/20 0.45
PNP P00491 1/20 0.45
MAPT P10636 1/20 0.45
DAO P14920 1/20 0.45
TSHR P16473 1/20 0.41
KDM4C Q9H3R0 2/20 0.40
SMN1; SMN2 Q16637 2/20 0.40
CYP1A2 P05177 2/20 0.40
CYP2C19 P33261 2/20 0.40
NPC1 O15118 1/20 0.40
RAB9A P51151 1/20 0.40
ALDH1A1 P00352 2/20 0.39
PTPRA P18433 1/20 0.39
KDM6B O15054 1/20 0.39
KDM4A O75164 1/20 0.39
KDM5C P41229 1/20 0.39
KDM2A Q9Y2K7 1/20 0.39
KDM3A Q9Y4C1 1/20 0.39
HRH4 Q9H3N8 1/20 0.38
HRH3 Q9Y5N1 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14604111 0.80 GAA (0.45) KDM4EDAOTSHRSMN1; SMN2RAB9A
SCHEMBL14273024 0.76 RAB9A (0.46) KDM4EMAPTKDM4CSMN1; SMN2CYP1A2
SCHEMBL4649050 0.76 PNP (0.42) PNPDAOALDH1A1L3MBTL1
SCHEMBL7262256 0.75 PDE3B (0.47) KDM4EPNPMAPTDAOKDM4C
SCHEMBL31691416 0.72 KDM4E (0.45) KDM4EMAPTKDM4CSMN1; SMN2CYP1A2
SCHEMBL6472533 0.72 AKR1B1 (0.40) DAONPC1RAB9AALDH1A1L3MBTL1
SCHEMBL8829787 0.72 PNP (0.49) KDM4EPNPMAPTDAOTSHR
SCHEMBL6612453 0.71 HRH4 (0.42) KDM4ETSHRKDM4CSMN1; SMN2CYP1A2
SCHEMBL16486420 0.71 TSHR (0.43) KDM4EDAOTSHRKDM4CCYP1A2
SCHEMBL4969020 0.71 TSHR (0.42) KDM4EMAPTTSHRSMN1; SMN2CYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1960367-A2 SUBSTITUTED PYRAZOLE COMPOUNDS USEFUL AS SOLUBLE EPOXIDE HYDROLASE INHIBITORS Boehringer Ingelheim International GmbH (DE) 2008-08-27 EP disclosed
WO-2007067836-A2 SUBSTITUTED PYRAZOLE COMPOUNDS USEFUL AS SOLUBLE EPOXIDE HYDROLASE INHIBITORS BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2007-06-14 WO disclosed