SCHEMBL4649211

SCHEMBL4649211

COc1cccc(Cc2cc(F)c3[nH]cc(C(=O)O)c(=O)c3c2)c1

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.49
HPGD P15428 2/20 0.49
KDM4E B2RXH2 1/20 0.49
GUSB P08236 4/20 0.47
KDM4C Q9H3R0 1/20 0.45
KDM5B Q9UGL1 1/20 0.45
LMNA P02545 1/20 0.43
GABRA1 P14867 3/20 0.42
GABRB2 P47870 3/20 0.42
RAB9A P51151 2/20 0.42
GABRB1 P18505 2/20 0.42
GABRA3 P34903 2/20 0.42
MDH2 P40926 1/20 0.42
SMN1; SMN2 Q16637 1/20 0.42
MEN1 O00255 1/20 0.42
NPC1 O15118 1/20 0.42
KMT2A Q03164 1/20 0.42
GABRP O00591 1/20 0.41
GABRD O14764 1/20 0.41
GABRG2 P18507 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4649998 0.89 RAB9A (0.41) ALDH1A1HPGDKDM4ELMNAGABRA1
SCHEMBL4650809 0.88 PRKAB2 (0.47) ALDH1A1HPGDKDM4EGUSBKDM5B
SCHEMBL4650110 0.88 KDM5A (0.42) ALDH1A1HPGDKDM4EKDM4CKDM5B
SCHEMBL4649447 0.85 RAB9A (0.49) ALDH1A1HPGDKDM4ELMNAGABRA1
SCHEMBL4650041 0.83 ALDH1A1 (0.47) ALDH1A1HPGDKDM4EKDM5BLMNA
SCHEMBL4650022 0.82 ALDH1A1 (0.50) ALDH1A1HPGDKDM4ELMNAGABRA1
SCHEMBL4650046 0.81 RAB9A (0.47) ALDH1A1HPGDKDM4EGUSBLMNA
SCHEMBL4650793 0.81 ALDH1A1 (0.46) ALDH1A1HPGDKDM4ELMNAGABRA1
SCHEMBL4650011 0.80 KDM4C (0.45) ALDH1A1HPGDKDM4EGUSBKDM4C
SCHEMBL4650045 0.80 ALDH1A1 (0.46) ALDH1A1HPGDKDM4EGUSBLMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1963271-A1 QUINOLONE M1 RECEPTOR POSITIVE ALLOSTERIC MODULATORS Merck & Co., Inc. (US) 2008-09-03 EP claimed
WO-2007067489-A1 QUINOLONE M1 RECEPTOR POSITIVE ALLOSTERIC MODULATORS MERCK & CO., INC. (US) 2007-06-14 WO claimed
EP-1963271-A1 QUINOLONE M1 RECEPTOR POSITIVE ALLOSTERIC MODULATORS Merck & Co., Inc. (US) 2008-09-03 EP disclosed
WO-2007067489-A1 QUINOLONE M1 RECEPTOR POSITIVE ALLOSTERIC MODULATORS MERCK & CO., INC. (US) 2007-06-14 WO disclosed