SCHEMBL4650809

SCHEMBL4650809

COc1ccc(Cc2cc(F)c3[nH]cc(C(=O)O)c(=O)c3c2)cc1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PRKAB2 O43741 2/20 0.47
PRKAG1 P54619 2/20 0.47
PRKAA2 P54646 2/20 0.47
PRKAA1 Q13131 2/20 0.47
PRKAG3 Q9UGI9 2/20 0.47
PRKAG2 Q9UGJ0 2/20 0.47
PRKAB1 Q9Y478 2/20 0.47
ALDH1A1 P00352 3/20 0.46
HPGD P15428 2/20 0.46
KDM4E B2RXH2 1/20 0.46
LMNA P02545 1/20 0.45
GUSB P08236 2/20 0.44
CHRM1 P11229 2/20 0.43
KDM5A P29375 1/20 0.43
KDM5B Q9UGL1 1/20 0.43
HTT P42858 1/20 0.42
GABRA1 P14867 2/20 0.42
GABRB2 P47870 2/20 0.42
GABRB1 P18505 1/20 0.42
GABRA3 P34903 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4649211 0.88 ALDH1A1 (0.49) ALDH1A1HPGDKDM4ELMNAGUSB
SCHEMBL4649996 0.87 GABRA1 (0.56) ALDH1A1KDM4ELMNAGABRA1GABRB2
SCHEMBL4649442 0.87 ALDH1A1 (0.41) ALDH1A1HPGDKDM4ELMNAHTT
SCHEMBL4649277 0.87 ALDH1A1 (0.41) ALDH1A1HPGDKDM4ELMNAGABRA1
SCHEMBL4650041 0.86 ALDH1A1 (0.47) PRKAB2PRKAG1PRKAA2PRKAA1PRKAG3
SCHEMBL4649447 0.86 RAB9A (0.49) ALDH1A1HPGDKDM4ELMNAGABRA1
SCHEMBL4650793 0.83 ALDH1A1 (0.46) PRKAB2PRKAG1PRKAA2PRKAA1PRKAG3
SCHEMBL4349605 0.83 PRKAG1 (0.47) PRKAB2PRKAG1PRKAA2PRKAA1PRKAG3
SCHEMBL4650802 0.83 ALDH1A1 (0.53) ALDH1A1HPGDKDM4ELMNAKDM5A
SCHEMBL4650045 0.83 ALDH1A1 (0.46) ALDH1A1HPGDKDM4ELMNAGUSB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1963271-A1 QUINOLONE M1 RECEPTOR POSITIVE ALLOSTERIC MODULATORS Merck & Co., Inc. (US) 2008-09-03 EP claimed
WO-2007067489-A1 QUINOLONE M1 RECEPTOR POSITIVE ALLOSTERIC MODULATORS MERCK & CO., INC. (US) 2007-06-14 WO claimed
EP-1963271-A1 QUINOLONE M1 RECEPTOR POSITIVE ALLOSTERIC MODULATORS Merck & Co., Inc. (US) 2008-09-03 EP disclosed
WO-2007100366-A2 QUINOLONE M1 RECEPTOR POSITIVE ALLOSTERIC MODULATORS MERCK & CO., INC. (US) 2007-09-07 WO disclosed
WO-2007067489-A1 QUINOLONE M1 RECEPTOR POSITIVE ALLOSTERIC MODULATORS MERCK & CO., INC. (US) 2007-06-14 WO disclosed