SCHEMBL4649998

SCHEMBL4649998

O=C(O)c1c[nH]c2c(F)cc(Cc3cccc(OC(F)F)c3)cc2c1=O

nearest known ligand 0.41

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
RAB9A P51151 1/20 0.41
ALDH1A1 P00352 3/20 0.41
HPGD P15428 2/20 0.41
MDH2 P40926 1/20 0.41
SMN1; SMN2 Q16637 1/20 0.41
KDM4E B2RXH2 2/20 0.41
DAO P14920 2/20 0.40
LMNA P02545 1/20 0.40
GABRA1 P14867 2/20 0.39
GABRB2 P47870 2/20 0.39
GABRB1 P18505 1/20 0.39
GABRA3 P34903 1/20 0.39
CSNK2A2 P19784 1/20 0.38
CSNK2B P67870 1/20 0.38
CSNK2A1 P68400 1/20 0.38
CYP1A2 P05177 1/20 0.38
HSD17B10 Q99714 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4649442 0.90 ALDH1A1 (0.41) ALDH1A1HPGDMDH2SMN1; SMN2KDM4E
SCHEMBL4650110 0.89 KDM5A (0.42) RAB9AALDH1A1HPGDMDH2SMN1; SMN2
SCHEMBL4649211 0.89 ALDH1A1 (0.49) RAB9AALDH1A1HPGDMDH2SMN1; SMN2
SCHEMBL4649447 0.85 RAB9A (0.49) RAB9AALDH1A1HPGDMDH2SMN1; SMN2
SCHEMBL4650041 0.82 ALDH1A1 (0.47) RAB9AALDH1A1HPGDKDM4ELMNA
SCHEMBL4650022 0.81 ALDH1A1 (0.50) RAB9AALDH1A1HPGDKDM4EDAO
SCHEMBL4650046 0.80 RAB9A (0.47) RAB9AALDH1A1HPGDMDH2SMN1; SMN2
SCHEMBL4650793 0.80 ALDH1A1 (0.46) RAB9AALDH1A1HPGDMDH2SMN1; SMN2
SCHEMBL4650809 0.79 PRKAB2 (0.47) ALDH1A1HPGDMDH2SMN1; SMN2KDM4E
SCHEMBL4650139 0.79 ALDH1A1 (0.51) RAB9AALDH1A1HPGDMDH2SMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1963271-A1 QUINOLONE M1 RECEPTOR POSITIVE ALLOSTERIC MODULATORS Merck & Co., Inc. (US) 2008-09-03 EP disclosed
WO-2007067489-A1 QUINOLONE M1 RECEPTOR POSITIVE ALLOSTERIC MODULATORS MERCK & CO., INC. (US) 2007-06-14 WO disclosed