SCHEMBL4656017

SCHEMBL4656017

COCCONS(=O)(=O)c1sc(C)cc1C

nearest known ligand 0.36

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
FBP1 P09467 10/20 0.36
CREBBP Q92793 1/20 0.35
ALDH1A1 P00352 3/20 0.33
HTT P42858 3/20 0.32
CA2 P00918 3/20 0.32
LMNA P02545 3/20 0.32
MAPK1 P28482 1/20 0.31
HPGD P15428 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3923958 0.75 LMNA (0.40) ALDH1A1HTTCA2LMNAMAPK1
SCHEMBL2618496 0.64 ALDH1A1 (0.50) ALDH1A1HTTLMNAMAPK1HPGD
SCHEMBL22508643 0.63 ALDH1A1 (0.41) ALDH1A1HTTLMNAMAPK1HPGD
SCHEMBL15220314 0.60 FBP1 (0.40) FBP1CREBBP
SCHEMBL16024140 0.59 FBP1 (0.34) FBP1CREBBP
SCHEMBL4789468 0.59 CA2 (0.46) CA2
SCHEMBL6568298 0.57 MAPK1 (0.64) ALDH1A1HTTCA2LMNAMAPK1
SCHEMBL266769 0.56 KDM1A (0.39) ALDH1A1HTTMAPK1HPGD
SCHEMBL28283415 0.54 TSHR (0.47) ALDH1A1CA2LMNAMAPK1HPGD
SCHEMBL12269650 0.53 PDE10A (0.31)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1996588-A1 NOVEL DUAL ACTION RECEPTORS ANTAGONISTS (DARA) AT THE ATI AND ETA RECEPTORS Torrent Pharmaceuticals Ltd (IN) 2008-12-03 EP disclosed
WO-2007100295-A1 NOVEL DUAL ACTION RECEPTORS ANTAGONISTS (DARA) AT THE ATI AND ETA RECEPTORS TORRENT PHARMACEUTICALS LTD (IN) 2007-09-07 WO disclosed