SCHEMBL4656444

SCHEMBL4656444

N#CC(C#N)(CCF)Cc1ccccc1Br

nearest known ligand 0.39

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
TAAR1 Q96RJ0 3/20 0.39
CYP1A1 P04798 1/20 0.36
CYP1A2 P05177 1/20 0.36
CYP1B1 Q16678 1/20 0.36
IDO1 P14902 2/20 0.34
PYCR1 P32322 1/20 0.32
SLC6A2 P23975 1/20 0.32
TSHR P16473 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28754249 0.75 TAAR1 (0.44) TAAR1CYP1A2IDO1PYCR1SLC6A2
SCHEMBL4657528 0.72 HTR2A (0.35) TAAR1CYP1A1CYP1A2CYP1B1IDO1
SCHEMBL14861015 0.72 TAAR1 (0.44) TAAR1CYP1A1CYP1A2CYP1B1IDO1
SCHEMBL30672075 0.72 TAAR1 (0.44) TAAR1CYP1A1CYP1A2CYP1B1IDO1
SCHEMBL4657538 0.71 TAAR1 (0.42) TAAR1CYP1A1CYP1A2CYP1B1IDO1
SCHEMBL263115 0.68 TAAR1 (0.46) TAAR1CYP1A2IDO1PYCR1SLC6A2
SCHEMBL4657442 0.67 LOXL2 (0.39) TAAR1IDO1
SCHEMBL4657455 0.67 TAAR1 (0.36) TAAR1IDO1
SCHEMBL4657492 0.66 IDO1 (0.36) TAAR1IDO1PYCR1
SCHEMBL4656045 0.66 SLC6A4 (0.40) TAAR1IDO1SLC6A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1385817-B1 MALONONITRILE COMPOUNDS AND THEIR USE AS PESTICIDES SUMITOMO CHEMICAL CO (JP) 2008-12-03 EP disclosed
US-7402691-B2 Malononitrile compounds and their use as pesticides SUMITOMO CHEMICAL COMPANY, LIMITED (JP) 2008-07-22 US disclosed
US-7011838-B2 Malononitrile compounds and their use as pesticides SUMITOMO CHEMICAL COMPANY, LIMITED (JP) 2006-03-14 US disclosed
US-20050209323-A1 Malononitrile compounds and their use as pesticides OTAKA KEN 2005-09-22 US disclosed
US-20040138065-A1 Malononitrile compounds and their use as pesticides SUMITOMO CHEMICAL COMPANY, LIMITED (JP) 2004-07-15 US disclosed
EP-1385817-A2 MALONONITRILE COMPOUNDS AND THEIR USE AS PESTICIDES SUMITOMO CHEMICAL COMPANY LIMITED (JP) 2004-02-04 EP disclosed
WO-2002090320-A2 MALONONITRILE COMPOUNDS AND THEIR USE AS PESTICIDES SUMITOMO CHEMICAL COMPANY, LIMITED (JP) 2002-11-14 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20050209323-A1 Malononitrile compounds and their use as pesticides C1S, C1R, C5 TAAR1 644/4885CYP1A1 280/4885CYP1A2 700/4885
US-20040138065-A1 Malononitrile compounds and their use as pesticides CBR1, MAL2, CBR3 TAAR1 632/4885CYP1A1 135/4885CYP1A2 642/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.