SCHEMBL4657455

SCHEMBL4657455

N#CC(C#N)(CCC(F)(F)F)Cc1ccccc1F

nearest known ligand 0.36

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
TAAR1 Q96RJ0 3/20 0.36
IDO1 P14902 2/20 0.34
ALDH1A1 P00352 3/20 0.34
KMT2A Q03164 2/20 0.34
POLB P06746 1/20 0.34
L3MBTL1 Q9Y468 4/20 0.33
LMNA P02545 3/20 0.33
TDP1 Q9NUW8 2/20 0.33
PKM P14618 2/20 0.33
MAPT P10636 3/20 0.31
AOC3 Q16853 1/20 0.31
NR3C1 P04150 1/20 0.30
NR3C2 P08235 1/20 0.30
MEN1 O00255 1/20 0.30
HTT P42858 1/20 0.30
ADORA2B P29275 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4657492 0.82 IDO1 (0.36) TAAR1IDO1ALDH1A1LMNAPKM
SCHEMBL4657490 0.81 IDO1 (0.38) IDO1NR3C1NR3C2
SCHEMBL4657447 0.77 ATM (0.40) TAAR1ALDH1A1LMNA
SCHEMBL11566464 0.73 TAAR1 (0.42) TAAR1IDO1ALDH1A1KMT2APOLB
SCHEMBL4658834 0.72 MAOA (0.33) TAAR1IDO1ALDH1A1KMT2A
SCHEMBL4657487 0.72 ALDH1A1 (0.33) ALDH1A1KMT2AMEN1HTT
SCHEMBL4657516 0.72 KDM4E (0.37) ALDH1A1KMT2APOLBL3MBTL1TDP1
SCHEMBL4657362 0.72 NR3C1 (0.37) ALDH1A1KMT2AL3MBTL1TDP1MAPT
SCHEMBL4658886 0.71
SCHEMBL4516471 0.71 KDM4E (0.36) ALDH1A1KMT2APOLBMAPTMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1385817-B1 MALONONITRILE COMPOUNDS AND THEIR USE AS PESTICIDES SUMITOMO CHEMICAL CO (JP) 2008-12-03 EP disclosed
US-7402691-B2 Malononitrile compounds and their use as pesticides SUMITOMO CHEMICAL COMPANY, LIMITED (JP) 2008-07-22 US disclosed
US-7011838-B2 Malononitrile compounds and their use as pesticides SUMITOMO CHEMICAL COMPANY, LIMITED (JP) 2006-03-14 US disclosed
US-20050209323-A1 Malononitrile compounds and their use as pesticides OTAKA KEN 2005-09-22 US disclosed
US-20040138065-A1 Malononitrile compounds and their use as pesticides SUMITOMO CHEMICAL COMPANY, LIMITED (JP) 2004-07-15 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20050209323-A1 Malononitrile compounds and their use as pesticides C1S, C1R, C5 TAAR1 644/4885IDO1 382/4885ALDH1A1 1502/4885
US-20040138065-A1 Malononitrile compounds and their use as pesticides CBR1, MAL2, CBR3 TAAR1 632/4885IDO1 278/4885ALDH1A1 614/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.