SCHEMBL4657516

SCHEMBL4657516

COc1cccc(CC(C#N)(C#N)CCC(F)(F)F)c1OC

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 4/20 0.37
TSHR P16473 2/20 0.37
ALOX15 P16050 1/20 0.37
TDP1 Q9NUW8 1/20 0.37
ALDH1A1 P00352 3/20 0.37
MAPK1 P28482 2/20 0.37
MEN1 O00255 2/20 0.37
KMT2A Q03164 2/20 0.37
HPGD P15428 1/20 0.37
ALOX12 P18054 1/20 0.37
CASP1 P29466 1/20 0.37
CASP7 P55210 1/20 0.37
ATM Q13315 1/20 0.37
NPSR1 Q6W5P4 1/20 0.37
HSD17B10 Q99714 1/20 0.37
AR P10275 1/20 0.37
ABCB1 P08183 3/20 0.36
GAA P10253 2/20 0.36
ABCG2 Q9UNQ0 1/20 0.36
CA12 O43570 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6824648 0.80 ALDH1A1 (0.43) KDM4ETSHRALDH1A1MAPK1MEN1
SCHEMBL11089198 0.74 CA12 (0.40) KDM4ETSHRALDH1A1MAPK1MEN1
SCHEMBL4657455 0.72 TAAR1 (0.36) TDP1ALDH1A1MEN1KMT2APOLB
SCHEMBL4658796 0.71 TAAR1 (0.42) MEN1KMT2AAR
SCHEMBL10190891 0.71 RIPK1 (0.49) KDM4ETSHRALDH1A1MAPK1MEN1
SCHEMBL4657492 0.71 IDO1 (0.36) KDM4EALDH1A1NPSR1
SCHEMBL27929732 0.70 SMN1; SMN2 (0.50) KDM4ETSHRALDH1A1MAPK1MEN1
SCHEMBL4657428 0.70 ALDH1A1 (0.39) TSHRALOX15ALDH1A1ALOX12AR
SCHEMBL4160051 0.70 SMN1; SMN2 (0.46) KDM4ETSHRALDH1A1MAPK1MEN1
SCHEMBL4761942 0.68 CA12 (0.48) KDM4ETSHRALDH1A1MAPK1MEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1385817-B1 MALONONITRILE COMPOUNDS AND THEIR USE AS PESTICIDES SUMITOMO CHEMICAL CO (JP) 2008-12-03 EP disclosed
US-7402691-B2 Malononitrile compounds and their use as pesticides SUMITOMO CHEMICAL COMPANY, LIMITED (JP) 2008-07-22 US disclosed
US-7011838-B2 Malononitrile compounds and their use as pesticides SUMITOMO CHEMICAL COMPANY, LIMITED (JP) 2006-03-14 US disclosed
US-20050209323-A1 Malononitrile compounds and their use as pesticides OTAKA KEN 2005-09-22 US disclosed
US-20040138065-A1 Malononitrile compounds and their use as pesticides SUMITOMO CHEMICAL COMPANY, LIMITED (JP) 2004-07-15 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20050209323-A1 Malononitrile compounds and their use as pesticides C1S, C1R, C5 KDM4E 1754/4885TSHR 2542/4885ALOX15 931/4885
US-20040138065-A1 Malononitrile compounds and their use as pesticides CBR1, MAL2, CBR3 KDM4E 1181/4885TSHR 3805/4885ALOX15 1802/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.