SCHEMBL4659945

SCHEMBL4659945

CCCCCC1=CCCC=C1c1ccccc1

nearest known ligand 0.41

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
GPR84 Q9NQS5 1/20 0.41
CNR1 P21554 2/20 0.40
CNR2 P34972 1/20 0.40
GAA P10253 1/20 0.40
HTT P42858 1/20 0.40
HSD11B1 P28845 1/20 0.40
TSHR P16473 1/20 0.38
PTPN1 P18031 2/20 0.37
DHFR P00374 1/20 0.37
GCGR P47871 2/20 0.36
KCNH2 Q12809 1/20 0.36
TRPV1 Q8NER1 1/20 0.35
LIPG Q9Y5X9 1/20 0.35
SIGMAR1 Q99720 1/20 0.35
MAPT P10636 2/20 0.35
TP53 P04637 1/20 0.35
SMN1; SMN2 Q16637 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4661287 0.98 CNR1 (0.40) GPR84CNR1CNR2GAAHTT
SCHEMBL4662723 0.95 TSHR (0.39) GPR84CNR1CNR2GAAHTT
Biphenyl SCHEMBL15347228 0.70 ALDH1A1 (0.56) GPR84GAAHTTHSD11B1TSHR
SCHEMBL13974896 0.69 PTPN1 (0.55) GPR84CNR1HSD11B1PTPN1
SCHEMBL19215836 0.68 PTGS2 (0.36) GPR84GAAHTTTSHRPTPN1
SCHEMBL5614129 0.68 SIGMAR1 (0.53) CNR1GAAHTTPTPN1SIGMAR1
Biphenyl SCHEMBL27853080 0.68 ALDH1A1 (0.53) GPR84HTTTSHRMAPTTP53
Biphenyl SCHEMBL5868587 0.68 ALDH1A1 (0.53) GPR84HTTTSHRMAPTTP53
Biphenyl SCHEMBL27342649 0.68 ALDH1A1 (0.53) GPR84HTTTSHRMAPTTP53
Hexadecane SCHEMBL8524813 0.68 ALDH1A1 (0.53) GPR84HTTTSHRMAPTTP53

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1919907-A2 HETEROCYCLIC COMPOUND OTSUKA PHARMACEUTICAL CO., LTD. (JP) 2008-05-14 EP disclosed
WO-2007026959-A2 DERIVATIVES OF 4-PIPERAZIN-1-YL-4-BENZ0 [B] THIOPHENE SUITABLE FOR THE TREATMENT OF CNS DISORDERS OTSUKA PHARMACEUTICAL CO., LTD. (JP) 2007-03-08 WO disclosed