SCHEMBL5614129

SCHEMBL5614129

CCCCCC1=CCCc2ccccc21

nearest known ligand 0.74

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
SIGMAR1 Q99720 4/20 0.53
GAA P10253 1/20 0.44
HTT P42858 1/20 0.44
PTPN1 P18031 1/20 0.43
CNR1 P21554 1/20 0.40
MPO P05164 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9235448 0.88 SIGMAR1 (0.50) SIGMAR1MPO
SCHEMBL2952166 0.86 SIGMAR1 (0.71) SIGMAR1
SCHEMBL29385038 0.83 HTR6 (0.46) SIGMAR1PTPN1CNR1
SCHEMBL16913235 0.83 HTR6 (0.46) SIGMAR1PTPN1CNR1
SCHEMBL14290594 0.81 SIGMAR1 (0.55) SIGMAR1
SCHEMBL11543020 0.81 SIGMAR1 (0.51) SIGMAR1CNR1
SCHEMBL11503302 0.80 MPO (0.57) SIGMAR1HTTMPO
SCHEMBL30151590 0.80 PTPN1 (0.43) SIGMAR1PTPN1CNR1
SCHEMBL7406702 0.77 SIGMAR1 (0.50) SIGMAR1MPO
SCHEMBL20430497 0.77 HTR6 (0.47) SIGMAR1PTPN1CNR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6608212-B1 Palladium catalyzed coupling of a vinylphosphate and aryl-metal halide; preparation of such as 1-(4-(2-(pyrrolidin-n-yl)-ethoxy)phenyl)-6-methoxy-3,4-dihydronaphthalene PFIZER, INC. 2003-08-19 US claimed
EP-1754709-A1 Process for preparing vinylphosphates DSM IP Assets B.V. (NL) 2007-02-21 EP disclosed
EP-1509484-A2 PROCESS FOR PREPARING VINYLAROMATIC COMPOUNDS DSM IP Assets B.V. (NL) 2005-03-02 EP disclosed
WO-2003102202-A2 PROCESS FOR PREPARING VINYLAROMATIC COMPOUNDS DSM IP ASSETS B.V. (NL) 2003-12-11 WO disclosed
US-6608212-B1 Palladium catalyzed coupling of a vinylphosphate and aryl-metal halide; preparation of such as 1-(4-(2-(pyrrolidin-n-yl)-ethoxy)phenyl)-6-methoxy-3,4-dihydronaphthalene PFIZER, INC. 2003-08-19 US disclosed