SCHEMBL4661396

SCHEMBL4661396

CCC(C#N)(C(=O)O)C(c1ccccc1C(C)C)c1cccc2ccccc12

nearest known ligand 0.38

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
PPARG P37231 1/20 0.38
PPARA Q07869 1/20 0.38
CYP2C9 P11712 2/20 0.37
CYP2C19 P33261 2/20 0.37
HPGD P15428 1/20 0.37
HTT P42858 1/20 0.37
LMNA P02545 1/20 0.37
GAA P10253 1/20 0.37
EPHX2 P34913 2/20 0.37
SLC6A4 P31645 1/20 0.36
ALOX5 P09917 1/20 0.36
CTSS P25774 1/20 0.35
CTSK P43235 1/20 0.35
ALDH1A1 P00352 1/20 0.35
ACP3 P15309 1/20 0.35
CYP1A2 P05177 1/20 0.35
PTGER4 P35408 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4662654 0.88 PPARG (0.38) PPARGPPARACYP2C9CYP2C19HPGD
SCHEMBL4661587 0.86 ESR1 (0.45) PPARGPPARAHPGDHTTGAA
SCHEMBL4661407 0.86 PPARG (0.46) PPARGPPARACYP2C9CYP2C19HPGD
SCHEMBL4661534 0.85 CMA1 (0.39) PPARGPPARACYP2C9CYP2C19HPGD
SCHEMBL4660153 0.85 PPARG (0.36) PPARGPPARACYP2C9CYP2C19HPGD
SCHEMBL4660128 0.83 ACP3 (0.42) PPARGPPARACYP2C9CYP2C19HPGD
SCHEMBL4660186 0.83 PPARG (0.37) PPARGPPARACYP2C9CYP2C19HPGD
SCHEMBL4661474 0.83 ALDH1A1 (0.42) PPARGPPARAGAAALDH1A1CYP1A2
SCHEMBL4661280 0.82 ESR1 (0.42) CYP2C9CYP2C19LMNAGAAALOX5
SCHEMBL6407531 0.82 ESR1 (0.42) CYP2C9CYP2C19LMNAGAAALOX5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1620102-B1 3-(1-NAPHTHYL)-2-CYANOPROPANOIC ACID DERIVATIVES AS ESTROGEN RECEPTOR LIGANDS WYETH CORP (US) 2008-12-24 EP claimed