SCHEMBL4661407

SCHEMBL4661407

CCC(C#N)(C(=O)O)C(c1ccccc1-c1ccccc1)c1cccc2ccccc12

nearest known ligand 0.46

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
PPARG P37231 10/20 0.46
PPARA Q07869 10/20 0.46
CYP2C9 P11712 3/20 0.44
CYP2C19 P33261 3/20 0.44
CYP1A2 P05177 1/20 0.44
PPARD Q03181 1/20 0.39
ACP3 P15309 2/20 0.37
ALOX5 P09917 1/20 0.37
CTSS P25774 1/20 0.36
CTSK P43235 1/20 0.36
CHRNB2 P17787 2/20 0.36
CHRNA4 P43681 2/20 0.36
CHRNB4 P30926 1/20 0.36
CHRNA3 P32297 1/20 0.36
HPGD P15428 1/20 0.36
HTT P42858 1/20 0.36
HDAC8 Q9BY41 1/20 0.35
HDAC6 Q9UBN7 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4660128 0.86 ACP3 (0.42) PPARGPPARACYP2C9CYP2C19CYP1A2
SCHEMBL4661396 0.86 PPARG (0.38) PPARGPPARACYP2C9CYP2C19CYP1A2
SCHEMBL4662654 0.86 PPARG (0.38) PPARGPPARACYP2C9CYP2C19CYP1A2
SCHEMBL4661587 0.84 ESR1 (0.45) PPARGPPARACTSSCTSKHPGD
SCHEMBL4660153 0.83 PPARG (0.36) PPARGPPARACYP2C9CYP2C19CYP1A2
SCHEMBL4660186 0.81 PPARG (0.37) PPARGPPARACYP2C9CYP2C19ACP3
SCHEMBL4661474 0.81 ALDH1A1 (0.42) PPARGPPARACYP1A2
SCHEMBL4661534 0.81 CMA1 (0.39) PPARGPPARACYP2C9CYP2C19ACP3
SCHEMBL4660080 0.80 ESR1 (0.42) PPARGPPARAHPGDHTT
SCHEMBL4661436 0.80 MEN1 (0.36) PPARGPPARACYP2C9CYP2C19CTSS

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1620102-B1 3-(1-NAPHTHYL)-2-CYANOPROPANOIC ACID DERIVATIVES AS ESTROGEN RECEPTOR LIGANDS WYETH CORP (US) 2008-12-24 EP claimed