SCHEMBL4661765

SCHEMBL4661765

CCCC1=CCCC=C1c1ccccc1

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CTSK P43235 1/20 0.35
HPGD P15428 4/20 0.33
KDM4E B2RXH2 3/20 0.33
ALDH1A1 P00352 3/20 0.33
SMN1; SMN2 Q16637 3/20 0.33
NPC1 O15118 2/20 0.33
RAB9A P51151 2/20 0.33
HSD17B10 Q99714 2/20 0.33
TSHR P16473 1/20 0.33
MAPT P10636 1/20 0.33
PKM P14618 1/20 0.33
ADORA1 P30542 3/20 0.33
ADORA3 P0DMS8 2/20 0.33
ADORA2A P29274 2/20 0.33
GAA P10253 1/20 0.32
SREBF2 Q12772 1/20 0.31
L3MBTL1 Q9Y468 1/20 0.31
PPARG P37231 1/20 0.31
TP53 P04637 1/20 0.31
TAAR1 Q96RJ0 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4662723 0.89 TSHR (0.39) TSHRADORA1GAA
SCHEMBL4659945 0.87 GPR84 (0.41) SMN1; SMN2TSHRMAPTGAATP53
SCHEMBL4661287 0.86 CNR1 (0.40) TSHRMAPTGAA
SCHEMBL28854031 0.69 ALDH1A1 (0.36) ALDH1A1TSHRL3MBTL1TAAR1
SCHEMBL5679087 0.66
SCHEMBL12992395 0.64 HSD17B10 (0.39) HPGDKDM4EALDH1A1SMN1; SMN2HSD17B10
SCHEMBL27975915 0.64 ALDH1A1 (0.47) CTSKHPGDKDM4EALDH1A1SMN1; SMN2
SCHEMBL9235448 0.64 SIGMAR1 (0.50)
SCHEMBL27365101 0.64 BACE1 (0.38) KDM4EALDH1A1NPC1RAB9ATSHR
Biphenyl SCHEMBL967556 0.63 ALDH1A1 (0.64) HPGDKDM4EALDH1A1SMN1; SMN2NPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1919907-A2 HETEROCYCLIC COMPOUND OTSUKA PHARMACEUTICAL CO., LTD. (JP) 2008-05-14 EP disclosed
WO-2007026959-A2 DERIVATIVES OF 4-PIPERAZIN-1-YL-4-BENZ0 [B] THIOPHENE SUITABLE FOR THE TREATMENT OF CNS DISORDERS OTSUKA PHARMACEUTICAL CO., LTD. (JP) 2007-03-08 WO disclosed