SCHEMBL4662728

SCHEMBL4662728

CC(O)c1ccccc1N(C)Cc1ccc(Br)nc1

nearest known ligand 0.48

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
MMP2 P08253 3/20 0.43
MMP9 P14780 3/20 0.43
MMP8 P22894 3/20 0.43
MMP13 P45452 3/20 0.43
CYP11B1 P15538 1/20 0.33
AOC3 Q16853 1/20 0.32
NPC1 O15118 2/20 0.31
RAB9A P51151 2/20 0.31
ALDH1A1 P00352 2/20 0.31
LMNA P02545 1/20 0.31
SMN1; SMN2 Q16637 1/20 0.31
KDM4E B2RXH2 1/20 0.31
KCNH2 Q12809 1/20 0.31
HDAC1 Q13547 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4661305 0.82 PYCR1 (0.42) NPC1ALDH1A1LMNASMN1; SMN2KDM4E
SCHEMBL4661399 0.82 PYCR1 (0.42) NPC1ALDH1A1LMNASMN1; SMN2KDM4E
SCHEMBL4661365 0.79 ACACB (0.43) MMP2MMP13
SCHEMBL4662731 0.76 PTPN1 (0.34) MMP2MMP9MMP8MMP13CYP11B1
SCHEMBL4662702 0.76 JAK2 (0.42) AOC3RAB9A
SCHEMBL4661242 0.73 POLB (0.45) LMNASMN1; SMN2KDM4E
SCHEMBL4661323 0.73 ALDH1A1 (0.41) MMP2MMP9MMP8MMP13ALDH1A1
SCHEMBL4661500 0.73 ALDH1A1 (0.41) MMP2MMP9MMP8MMP13ALDH1A1
SCHEMBL4664189 0.72 TYMS (0.46) MMP2MMP9MMP8MMP13ALDH1A1
SCHEMBL4346767 0.72 MEN1 (0.55) AOC3RAB9AALDH1A1LMNASMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2007707-A1 COMPOUNDS WHICH MODULATE THE CB2 RECEPTOR Boehringer Ingelheim International GmbH (DE) 2008-12-31 EP disclosed
WO-2007118041-A1 COMPOUNDS WHICH MODULATE THE CB2 RECEPTOR BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2007-10-18 WO disclosed