SCHEMBL4661365

SCHEMBL4661365

C[C@H](O)c1ccccc1N(C)Cc1ccc(Oc2ccccc2)nc1

nearest known ligand 0.43

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
ACACB O00763 9/20 0.43
GRN P28799 2/20 0.41
SORT1 Q99523 2/20 0.41
ACACA Q13085 5/20 0.40
CTSA P10619 2/20 0.39
LIPE Q05469 1/20 0.39
OPRM1 P35372 3/20 0.37
OPRD1 P41143 3/20 0.37
HRH3 Q9Y5N1 1/20 0.37
ADAMTS4 O75173 1/20 0.36
MMP1 P03956 1/20 0.36
MMP2 P08253 1/20 0.36
MMP13 P45452 1/20 0.36
MMP14 P50281 1/20 0.36
ADAMTS5 Q9UNA0 1/20 0.36
OPRK1 P41145 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4662728 0.79 MMP2 (0.43) MMP2MMP13
SCHEMBL4661367 0.79 ACACB (0.42) ACACBGRNSORT1ACACALIPE
SCHEMBL4342586 0.76 MEN1 (0.51) ACACBGRNSORT1LIPE
SCHEMBL4661336 0.75 ACACB (0.43) ACACBGRNSORT1ACACACTSA
SCHEMBL12844619 0.72 GRN (0.47) ACACBGRNSORT1OPRM1OPRD1
SCHEMBL4661305 0.72 PYCR1 (0.42)
SCHEMBL4661399 0.72 PYCR1 (0.42)
SCHEMBL12775823 0.71 ACACB (0.50) ACACBGRNSORT1ACACAOPRM1
SCHEMBL4662702 0.71 JAK2 (0.42)
SCHEMBL4661323 0.71 ALDH1A1 (0.41) MMP2MMP13

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2007707-A1 COMPOUNDS WHICH MODULATE THE CB2 RECEPTOR Boehringer Ingelheim International GmbH (DE) 2008-12-31 EP claimed
WO-2007118041-A1 COMPOUNDS WHICH MODULATE THE CB2 RECEPTOR BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2007-10-18 WO claimed
EP-2007707-A1 COMPOUNDS WHICH MODULATE THE CB2 RECEPTOR Boehringer Ingelheim International GmbH (DE) 2008-12-31 EP disclosed
WO-2007118041-A1 COMPOUNDS WHICH MODULATE THE CB2 RECEPTOR BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2007-10-18 WO disclosed