SCHEMBL4663041

SCHEMBL4663041

CSc1ccc(-c2ccccc2)c(C(F)(F)F)c1

nearest known ligand 0.41

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
S1PR1 P21453 6/20 0.41
S1PR3 Q99500 4/20 0.41
KDM4E B2RXH2 1/20 0.40
ALDH1A1 P00352 1/20 0.40
TDP1 Q9NUW8 1/20 0.40
L3MBTL1 Q9Y468 1/20 0.40
AKR1C3 P42330 4/20 0.38
AKR1C2 P52895 4/20 0.38
STK10 O94804 2/20 0.38
SLK Q9H2G2 2/20 0.38
PTGS2 P35354 1/20 0.38
RORC P51449 1/20 0.38
ESR2 Q92731 1/20 0.37
ACP1 P24666 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4663035 0.83 S1PR1 (0.41) S1PR1S1PR3AKR1C3AKR1C2RORC
SCHEMBL19086307 0.77 PTGS2 (0.41) AKR1C3AKR1C2PTGS2ESR2
SCHEMBL4637120 0.77 AKR1C3 (0.51) S1PR1S1PR3AKR1C3AKR1C2RORC
SCHEMBL27638533 0.76 S1PR1 (0.52) S1PR1S1PR3L3MBTL1AKR1C3AKR1C2
SCHEMBL4781603 0.74 KIF11 (0.54) S1PR1S1PR3ALDH1A1
SCHEMBL3578278 0.74 AR (0.40)
SCHEMBL4664565 0.73 RORC (0.38) S1PR1S1PR3KDM4EALDH1A1L3MBTL1
SCHEMBL30608015 0.73 KDM4E (0.44) KDM4EAKR1C3AKR1C2STK10SLK
SCHEMBL2942635 0.73 S1PR1 (0.47) S1PR1S1PR3ALDH1A1AKR1C3AKR1C2
SCHEMBL19259678 0.73 PTGS2 (0.41) AKR1C3AKR1C2PTGS2ESR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1638551-A4 IMMUNOSUPPRESSANT COMPOUNDS AND COMPOSITIONS IRM LLC (BM) 2008-12-31 EP disclosed
EP-1638551-A2 IMMUNOSUPPRESSANT COMPOUNDS AND COMPOSITIONS IRM LLC (BM) 2006-03-29 EP disclosed
WO-2004103309-A2 IMMUNOSUPPRESSANT COMPOUNDS AND COMPOSITIONS IRM LLC (BM) 2004-12-02 WO disclosed