SCHEMBL4664786

SCHEMBL4664786

CC(C)COC(=O)N1CC=C(c2c[nH]c3c(C#N)nc(-c4ccccc4)cc23)CC1

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
BTK Q06187 5/20 0.39
CHEK1 O14757 2/20 0.37
MAP4K4 O95819 2/20 0.37
CHEK2 O96017 2/20 0.37
PRKCG P05129 2/20 0.37
CDK1 P06493 2/20 0.37
PIM1 P11309 2/20 0.37
FGFR1 P11362 2/20 0.37
PRKACA P17612 2/20 0.37
RPS6KB1 P23443 2/20 0.37
CDK2 P24941 2/20 0.37
MARK3 P27448 2/20 0.37
MAPK1 P28482 2/20 0.37
FLT4 P35916 2/20 0.37
FLT3 P36888 2/20 0.37
CLK2 P49760 2/20 0.37
GSK3A P49840 2/20 0.37
GSK3B P49841 2/20 0.37
IRAK1 P51617 2/20 0.37
RPS6KA3 P51812 2/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4664978 0.88 BTK (0.40) BTKCHEK1MAP4K4CHEK2PRKCG
SCHEMBL4665003 0.87 JAK2 (0.38) BTKCHEK1MAP4K4CHEK2PRKCG
SCHEMBL4663355 0.86 JAK1 (0.46) BTKJAK1
SCHEMBL3715658 0.75 DRD2 (0.49) CHEK1MAP4K4CHEK2PRKCGCDK1
SCHEMBL4665049 0.74 JAK1 (0.48) BTKJAK1
SCHEMBL5007703 0.73 JAK1 (0.47) BTKJAK1
SCHEMBL4590003 0.72 WDR5 (0.40) BTKCHEK1MAP4K4CHEK2PRKCG
SCHEMBL5302846 0.69 IKBKB (0.43) MAPTJAK2JAK1LNPEPTDP1
SCHEMBL4666734 0.66 IKBKB (0.48) BTKFLT3AURKAJAK2
SCHEMBL3226626 0.66 MAPT (0.66) MAPTHTR1ADRD2TP53

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1940296-A2 CHEMICAL COMPOUNDS SmithKline Beecham Corporation (US) 2008-07-09 EP disclosed
WO-2007114848-A2 CHEMICAL COMPOUNDS SMITHKLINE BEECHAM CORPORATION (US) 2007-10-11 WO disclosed