SCHEMBL4667248

SCHEMBL4667248

C=CC1(O)CCC(Cc2ccc(Cl)cc2)CC1C(C)(C)N

nearest known ligand 0.36

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
TRPA1 O75762 2/20 0.36
SLC6A2 P23975 1/20 0.33
HTR2A P28223 1/20 0.33
SLC6A4 P31645 1/20 0.33
HRH1 P35367 1/20 0.33
HTR2B P41595 1/20 0.33
CHRNA4 P43681 1/20 0.33
SLC6A3 Q01959 1/20 0.33
ALDH1A1 P00352 1/20 0.32
CCR5 P51681 1/20 0.32
BCL2A1 Q16548 1/20 0.31
FPR2 P25090 1/20 0.30
PROKR1 Q8TCW9 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4665614 0.77 OPRM1 (0.35) TRPA1SLC6A2SLC6A4SLC6A3ALDH1A1
SCHEMBL4663768 0.65 TRPA1 (0.40) TRPA1SLC6A2SLC6A4SLC6A3
SCHEMBL4667249 0.63 TRPA1 (0.38) TRPA1CCR5
SCHEMBL29693296 0.62 ALDH1A1 (0.43) TRPA1ALDH1A1CCR5FPR2PROKR1
SCHEMBL4663731 0.62 OPRM1 (0.36) TRPA1SLC6A2SLC6A4SLC6A3ALDH1A1
SCHEMBL4665379 0.62 OPRK1 (0.42) SLC6A2SLC6A4SLC6A3ALDH1A1
SCHEMBL1119467 0.61 ALDH1A1 (0.59) SLC6A2SLC6A4ALDH1A1FPR2PROKR1
SCHEMBL4664004 0.60 SLC6A4 (0.37) TRPA1SLC6A2SLC6A4SLC6A3ALDH1A1
SCHEMBL4663567 0.60 SMN1; SMN2 (0.43) SLC6A2SLC6A4SLC6A3ALDH1A1
SCHEMBL4663513 0.60 SLC6A4 (0.36) TRPA1SLC6A2SLC6A4SLC6A3ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1571140-B1 C-substituted cyclohexylmethylamine derivatives GRUENENTHAL GMBH (DE) 2008-11-12 EP claimed