SCHEMBL4667518

SCHEMBL4667518

CCc1cc(Nc2ccc(Cl)cc2C(=O)OC)n(-c2ccncc2)n1

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KCNMA1 Q12791 1/20 0.39
ALDH1A1 P00352 3/20 0.39
KMT2A Q03164 3/20 0.39
MEN1 O00255 2/20 0.39
KDM4E B2RXH2 1/20 0.39
HPGD P15428 1/20 0.39
NPY1R P25929 1/20 0.39
NPY2R P49146 1/20 0.39
TGFBR1 P36897 1/20 0.38
GFER P55789 1/20 0.37
ABL1 P00519 1/20 0.36
TP53 P04637 1/20 0.36
RXFP1 Q9HBX9 1/20 0.36
LMNA P02545 3/20 0.35
CYP46A1 Q9Y6A2 1/20 0.35
NUDT1 P36639 1/20 0.35
MAPT P10636 3/20 0.35
CYP1A2 P05177 1/20 0.35
CYP2D6 P10635 1/20 0.35
CYP2C9 P11712 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4664665 0.85 TGFBR1 (0.40) KCNMA1ALDH1A1HPGDTGFBR1TP53
SCHEMBL4665548 0.83 ALDH1A1 (0.43) ALDH1A1KMT2AMEN1KDM4EHPGD
SCHEMBL27749269 0.83 TP53 (0.43) ALDH1A1KMT2AMEN1KDM4EHPGD
Hydrochloric Acid SCHEMBL27749272 0.82 TP53 (0.42) ALDH1A1KMT2AMEN1KDM4EHPGD
SCHEMBL4668860 0.79 KCNMA1 (0.38) KCNMA1ALDH1A1KMT2AMEN1KDM4E
SCHEMBL14600443 0.75 MAPK14 (0.53)
SCHEMBL14600709 0.73 MARS1 (0.43) ALDH1A1KMT2AMEN1KDM4ECYP1A2
SCHEMBL27728861 0.70 KMT2A (0.51) ALDH1A1KMT2AMEN1KDM4EHPGD
SCHEMBL15712337 0.69 KCNMA1 (0.41) KCNMA1KMT2AMEN1HPGDTGFBR1
SCHEMBL14600228 0.69 HPGD (0.38) ALDH1A1KMT2AMEN1KDM4EHPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1928455-A1 ANILINOPYRAZOLE DERIVATIVES USEFUL FOR THE TREATMENT OF DIABETES Bayer Healthcare, LLC (US) 2008-06-11 EP disclosed
WO-2007027842-A1 ANILINOPYRAZOLE DERIVATIVES USEFUL FOR THE TREATMENT OF DIABETES BAYER HEALTHCARE LLC (US) 2007-03-08 WO disclosed
WO-2007027842-A1 ANILINOPYRAZOLE DERIVATIVES USEFUL FOR THE TREATMENT OF DIABETES BAYER HEALTHCARE LLC (US) 2007-03-08 WO disclosed