SCHEMBL46717

SCHEMBL46717

O=C/C(=C/c1ccc(-c2ccc(Cl)c(C(=O)O)c2)o1)SC(=O)NCc1ccc(F)cc1

nearest known ligand 0.58

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 5/20 0.58
KDM4E B2RXH2 5/20 0.58
XPA P23025 2/20 0.49
KMT2A Q03164 9/20 0.49
MEN1 O00255 7/20 0.49
NPC1 O15118 3/20 0.49
RAB9A P51151 3/20 0.49
POLB P06746 5/20 0.44
TDP1 Q9NUW8 5/20 0.44
L3MBTL1 Q9Y468 4/20 0.44
APEX1 P27695 2/20 0.44
CTDSP1 Q9GZU7 2/20 0.44
DUSP26 Q9BV47 1/20 0.44
MAPT P10636 5/20 0.44
NPSR1 Q6W5P4 3/20 0.44
GAA P10253 2/20 0.44
HPGD P15428 1/20 0.44
ALOX12 P18054 1/20 0.44
TTR P02766 1/20 0.43
PKM P14618 3/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL46709 0.85 XPA (0.51) ALDH1A1KDM4EXPAKMT2AMEN1
SCHEMBL6721173 0.73 KDM4E (1.00) ALDH1A1KDM4EKMT2AMEN1NPC1
SCHEMBL19021491 0.72 ALDH1A1 (0.52) ALDH1A1KDM4EXPAKMT2AMEN1
SCHEMBL2556095 0.70 LDHA (0.72) ALDH1A1KDM4EKMT2AMEN1NPC1
SCHEMBL46199 0.70 XPA (0.48) ALDH1A1KDM4EXPAKMT2AMEN1
SCHEMBL6393879 0.70 TDP1 (0.74) ALDH1A1KDM4EKMT2AMEN1NPC1
SCHEMBL5146587 0.70 TDP1 (0.74) ALDH1A1KDM4EKMT2AMEN1NPC1
SCHEMBL46215 0.69 ENPP2 (0.75) ALDH1A1KDM4EKMT2AMEN1NPC1
SCHEMBL6721163 0.69 ALDH1A1 (0.75) ALDH1A1KDM4EKMT2AMEN1NPC1
SCHEMBL17789559 0.68 ALDH1A1 (0.53) ALDH1A1KDM4EXPAKMT2AMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012005800-A1 COMPOUNDS AND METHODS FOR REGULATING INTEGRIN CD11B/CD18 ADHAERE PHARAMACEUTICALS, INC. (US) 2012-01-12 WO disclosed