SCHEMBL4673189

SCHEMBL4673189

CCCC[CH]C(=O)CC(C)=O

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TSHR P16473 2/20 0.39
CES2 O00748 4/20 0.38
F7 P08709 1/20 0.36
F3 P13726 1/20 0.36
CES1 P23141 2/20 0.34
ALDH1A1 P00352 3/20 0.33
POLB P06746 3/20 0.33
TDP1 Q9NUW8 1/20 0.33
EP300 Q09472 1/20 0.33
POLA1 P09884 1/20 0.32
GMNN O75496 1/20 0.32
USP2 O75604 1/20 0.32
LMNA P02545 1/20 0.32
CYP1A2 P05177 1/20 0.32
MAPT P10636 1/20 0.32
CYP2C9 P11712 1/20 0.32
ALOX15 P16050 1/20 0.32
APEX1 P27695 1/20 0.32
CYP2C19 P33261 1/20 0.32
RECQL P46063 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL128203 0.78
SCHEMBL4091375 0.76
SCHEMBL129431 0.76 F7 (0.43) TSHRCES2F7F3CES1
SCHEMBL27322155 0.75
SCHEMBL125167 0.75
SCHEMBL3330873 0.74 TRPA1 (0.52) CES2F7F3CES1POLB
SCHEMBL13061577 0.73 EP300 (0.42) TSHRCES2F7F3CES1
SCHEMBL788432 0.73 CES2 (0.52) TSHRCES2F7F3CES1
SCHEMBL572485 0.73 CES2 (0.52) TSHRCES2F7F3CES1
SCHEMBL7180871 0.73 CES2 (0.52) TSHRCES2F7F3CES1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 14 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20060084590-A1 Methods of and compounds for modulating the activity of bacterial FabG SMITHKLINE BEECHAM CORPORATION 2006-04-20 US claimed
US-20050026187-A1 Methods of and compounds for modulating the activity of bacterial FabG SMITHKLINE BEECHAM CORPORATION 2005-02-03 US claimed
CN-103074308-B Enzyme of Cordyceps hirsutella sinensis for synthesis of 3-hydroxybutyrate, and gene and application thereof UNIV ZHEJIANG TECHNOLOGY 2014-06-11 CN disclosed
CN-103074308-B Enzyme of Cordyceps hirsutella sinensis for synthesis of 3-hydroxybutyrate, and gene and application thereof UNIV ZHEJIANG TECHNOLOGY 2014-06-11 CN disclosed
WO-2013130481-A1 RECOMBINANT HOST CELLS AND PROCESSES FOR PRODUCING 1,3-BUTADIENE THROUGH A CROTONOL INTERMEDIATE CODEXIS, INC. (US) 2013-09-06 WO disclosed
CN-103074308-A Enzyme of Cordyceps hirsutella sinensis for synthesis of 3-hydroxybutyrate, and gene and application thereof UNIV ZHEJIANG TECHNOLOGY 2013-05-01 CN disclosed
CN-103074308-A Enzyme of Cordyceps hirsutella sinensis for synthesis of 3-hydroxybutyrate, and gene and application thereof UNIV ZHEJIANG TECHNOLOGY 2013-05-01 CN disclosed
US-20080161247-A1 Synergistic composition for modulating activity of substrate analogs for NAD+, NADP+, NADH or NADPH dependent enzymes and process thereof NATIONAL INSTITUTE OF IMMUNOLOGY AND INDIAN INSTITUTE OF SCIENCE 2008-07-03 US disclosed
EP-1938841-A2 Synergistic composition for modulating activity of substrate analogs for NAD+, NADP+, NADH+ or NADPH dependent enzymes and process thereof National Institute of Immunology (IN) 2008-07-02 EP disclosed
US-20060084590-A1 Methods of and compounds for modulating the activity of bacterial FabG SMITHKLINE BEECHAM CORPORATION 2006-04-20 US disclosed
US-6881553-B2 Antimicrobial activity of gemfibrozil and related compounds and derivatives and metabolites thereof THE TRUSTEES OF COLUMBIA UNIVERSITY IN THE CITY OF NEW YORK (US) 2005-04-19 US disclosed
US-20050026187-A1 Methods of and compounds for modulating the activity of bacterial FabG SMITHKLINE BEECHAM CORPORATION 2005-02-03 US disclosed
US-20030191146-A1 Novel antimicrobial activity of gemfibrozil and related compounds and derivatives and metabolites thereof THE TRUSTEES OF COLUMBIA UNIVERSITY IN THE CITY OF NEW YORK 2003-10-09 US disclosed
US-6531291-B1 Which inhibit enoyl reductase; drug screening THE TRUSTEES OF COLUMBIA UNIVERSITY IN THE CITY OF NEW YORK 2003-03-11 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20080161247-A1 Synergistic composition for modulating activity of substrate analogs for NAD+, NADP+, NADH or NADPH dependent enzymes and process thereof NQO1, NADK, TECR TSHR 2794/4885CES2 2568/4885F7 4574/4885
US-20030191146-A1 Novel antimicrobial activity of gemfibrozil and related compounds and derivatives and metabolites thereof CBR1, CBR3, GCDH TSHR 889/4885CES2 89/4885F7 2248/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.