SCHEMBL4674989

SCHEMBL4674989

CCCNC(=O)c1ccc(-n2ccnc2)cc1

nearest known ligand 0.60

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 1/20 0.60
BAZ2B Q9UIF8 1/20 0.60
HTT P42858 1/20 0.59
CYP4Z1 Q86W10 1/20 0.57
DRD3 P35462 4/20 0.55
ADRB2 P07550 2/20 0.55
ADRB1 P08588 2/20 0.55
ADRB3 P13945 2/20 0.55
MAPT P10636 2/20 0.54
L3MBTL1 Q9Y468 1/20 0.54
TDP1 Q9NUW8 1/20 0.54
ADH5 P11766 1/20 0.54
DRD2 P14416 3/20 0.53
HTR2A P28223 1/20 0.51
HTR2C P28335 1/20 0.51
HTR2B P41595 1/20 0.51
KMT2A Q03164 2/20 0.51
GFER P55789 1/20 0.51
GAA P10253 1/20 0.50
MAOB P27338 1/20 0.50

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7068530 0.90 NAAA (0.63) CYP3A4BAZ2BHTTCYP4Z1DRD3
SCHEMBL9368933 0.89 CYP3A4 (0.63) CYP3A4BAZ2BHTTCYP4Z1DRD3
SCHEMBL9363661 0.87 ALDH1A1 (0.58) CYP3A4BAZ2BHTTCYP4Z1DRD3
SCHEMBL8781065 0.86 CYP4Z1 (0.57) CYP3A4BAZ2BHTTCYP4Z1DRD3
Hydrochloric Acid SCHEMBL9363955 0.86 BLM (0.59) CYP3A4BAZ2BHTTCYP4Z1DRD3
SCHEMBL9363643 0.85 DRD3 (0.51) CYP3A4BAZ2BHTTCYP4Z1DRD3
Hydrochloric Acid SCHEMBL8781047 0.85 CYP4Z1 (0.56) CYP3A4BAZ2BHTTCYP4Z1DRD3
SCHEMBL9363630 0.85 DRD3 (0.55) CYP3A4BAZ2BHTTCYP4Z1DRD3
Hydrochloric Acid SCHEMBL9364164 0.84 DRD3 (0.54) CYP3A4BAZ2BHTTCYP4Z1DRD3
SCHEMBL9369002 0.83 TDP1 (0.52) CYP3A4BAZ2BHTTCYP4Z1DRD3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1885697-A2 SOLUBLE EPOXIDE HYDROLASE INHIBITORS AND METHODS OF USING SAME BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2008-02-13 EP disclosed
WO-2006121719-A2 SOLUBLE EPOXIDE HYDROLASE INHIBITORS AND METHODS OF USING SAME BOEHRINGER INGELHEIM INTERNATIONAL, GMBH (DE) 2006-11-16 WO disclosed