SCHEMBL4682203

SCHEMBL4682203

[O]CCS(=O)(=O)c1ncc[nH]1

nearest known ligand 0.38

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
TAAR1 Q96RJ0 5/20 0.33
ALOX15 P16050 1/20 0.33
TXNRD1 Q16881 1/20 0.33
FDPS P14324 1/20 0.33
ALDH1A1 P00352 1/20 0.32
SMN1; SMN2 Q16637 1/20 0.32
TBXAS1 P24557 2/20 0.32
HTR1A P08908 1/20 0.32
PSEN1 P49768 1/20 0.31
PSEN2 P49810 1/20 0.31
APH1B Q8WW43 1/20 0.31
NCSTN Q92542 1/20 0.31
APH1A Q96BI3 1/20 0.31
PSENEN Q9NZ42 1/20 0.31
TERT O14746 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7288664 0.89 TBXAS1 (0.33) TAAR1ALOX15TXNRD1FDPSALDH1A1
SCHEMBL4681643 0.85 TBXAS1 (0.35) TAAR1ALOX15TXNRD1TBXAS1
SCHEMBL7296081 0.85 TBXAS1 (0.35) TAAR1ALOX15TXNRD1TBXAS1
SCHEMBL4686081 0.83 ALDH1A1 (0.34) TAAR1ALOX15TXNRD1FDPSALDH1A1
SCHEMBL4682206 0.82 CA2 (0.36) TAAR1ALOX15TXNRD1FDPSALDH1A1
SCHEMBL7288670 0.79 CA2 (0.40) TAAR1ALOX15TXNRD1FDPSTBXAS1
SCHEMBL2010779 0.79 ALDH1A1 (0.39) TAAR1ALOX15TXNRD1ALDH1A1SMN1; SMN2
SCHEMBL2851629 0.78 EPHX2 (0.39) TAAR1TXNRD1HTR1A
SCHEMBL4686083 0.78 TBXAS1 (0.36) ALOX15TXNRD1FDPSALDH1A1SMN1; SMN2
Hydrochloric Acid SCHEMBL4002548 0.77 TAAR1 (0.34) TAAR1ALOX15TXNRD1ALDH1A1SMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1902717-A2 Vasopressin antagonist and oxytocin antagonist Otsuka Pharmaceutical Company, Limited (JP) 2008-03-26 EP disclosed
EP-0620003-B1 VASOPRESSIN ANTAGONIST AND OXYTOCIN ANTAGONIST OTSUKA PHARMA CO LTD (JP) 2008-01-16 EP disclosed
US-5753644-A Vasopressin antagonist and oxytocin antagonist OTSUKA PHARMACEUTICAL CO., LTD. (JP) 1998-05-19 US disclosed
US-5622947-A VASODILATORS, HYPOTENSIVE AGENTS, DIURETICS, PLATELET AGGLUTINATION INHIBITORS; ALSO USED TO PREVENT PREMATURE BIRTH, TREAT DYSMENORRHEA OTSUKA PHARMACEUTICAL CO., LTD. (JP) 1997-04-22 US disclosed
EP-0620003-A1 VASOPRESSIN ANTAGONIST AND OXYTOCIN ANTAGONIST OTSUKA PHARMACEUTICAL CO., LTD. (JP) 1994-10-19 EP disclosed