SCHEMBL4686109

SCHEMBL4686109

OCCCCCSc1c[nH]cn1

nearest known ligand 0.35

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
CA2 P00918 3/20 0.35
GBA1 P04062 1/20 0.35
GSTP1 P09211 2/20 0.31
GSTM2 P28161 2/20 0.31
AURKA O14965 1/20 0.31
GPR84 Q9NQS5 1/20 0.30
KDM6B O15054 1/20 0.30
KDM4A O75164 1/20 0.30
KDM4D Q6B0I6 1/20 0.30
KDM3B Q7LBC6 1/20 0.30
HIF1AN Q9NWT6 1/20 0.30
KDM5B Q9UGL1 1/20 0.30
KDM2A Q9Y2K7 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7287495 0.98 CA2 (0.33) CA2GBA1GSTP1GSTM2
SCHEMBL9435821 0.78
SCHEMBL1052495 0.75 HPRT1 (0.35)
SCHEMBL4684788 0.68 ALDH1A1 (0.56)
SCHEMBL4685852 0.68 ALDH1A1 (0.56)
SCHEMBL4682895 0.67 PKM (0.42) CA2GSTP1GSTM2GPR84
SCHEMBL4685958 0.66 ALDH1A1 (0.49)
SCHEMBL4687627 0.66 ALDH1A1 (0.57)
SCHEMBL4686177 0.66 FDPS (0.50) CA2GPR84KDM6BKDM4AKDM4D
SCHEMBL7356738 0.66 FDPS (0.50) CA2GPR84KDM6BKDM4AKDM4D

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1902717-A2 Vasopressin antagonist and oxytocin antagonist Otsuka Pharmaceutical Company, Limited (JP) 2008-03-26 EP disclosed
EP-0620003-B1 VASOPRESSIN ANTAGONIST AND OXYTOCIN ANTAGONIST OTSUKA PHARMA CO LTD (JP) 2008-01-16 EP disclosed
US-5753644-A Vasopressin antagonist and oxytocin antagonist OTSUKA PHARMACEUTICAL CO., LTD. (JP) 1998-05-19 US disclosed
US-5622947-A VASODILATORS, HYPOTENSIVE AGENTS, DIURETICS, PLATELET AGGLUTINATION INHIBITORS; ALSO USED TO PREVENT PREMATURE BIRTH, TREAT DYSMENORRHEA OTSUKA PHARMACEUTICAL CO., LTD. (JP) 1997-04-22 US disclosed
EP-0620003-A1 VASOPRESSIN ANTAGONIST AND OXYTOCIN ANTAGONIST OTSUKA PHARMACEUTICAL CO., LTD. (JP) 1994-10-19 EP disclosed