SCHEMBL4687689

SCHEMBL4687689

COC(Cc1cc(C(=O)O)ccc1[N+](=O)[O-])OC

nearest known ligand 0.54

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
CASP6 P55212 1/20 0.54
TSHR P16473 2/20 0.54
POLB P06746 1/20 0.50
HCAR3 P49019 12/20 0.49
LMNA P02545 1/20 0.47
MAPT P10636 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4233674 0.82 HCAR3 (0.40) CASP6TSHRHCAR3LMNA
SCHEMBL4299408 0.81 CASP6 (0.58) CASP6TSHRPOLBHCAR3LMNA
SCHEMBL29897189 0.81 CASP6 (0.58) CASP6TSHRPOLBHCAR3LMNA
SCHEMBL1609806 0.81 CASP6 (0.66) CASP6TSHRPOLBHCAR3LMNA
Hydrochloric Acid SCHEMBL1609389 0.79 CASP6 (0.64) CASP6TSHRPOLBHCAR3LMNA
SCHEMBL4990608 0.78 KMT2A (0.49) TSHRPOLBLMNAMAPT
SCHEMBL2263152 0.78 ALOX15 (0.39) TSHRLMNAMAPT
SCHEMBL18027781 0.77 CASP6 (0.66) CASP6TSHRPOLBHCAR3LMNA
SCHEMBL544105 0.77 VCAM1 (0.54) POLBLMNA
SCHEMBL17399916 0.77 CASP6 (0.60) CASP6TSHRPOLBHCAR3LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1732887-B1 1-(1H-INDOL-1-YL)-3-(4-METHYLPIPERAZIN-1-YL)-1-PHENYL PROPAN-2-OL DERIVATIVES AND RELATED COMPOUNDS AS MODULATORS OF THE NOREPINEPHRINE (NE) AND THE SEROTONINE (5-HT) ACTIVITY AND THE MONOAMINE REUPTAKE FOR THE TREATMENT OF VASOMOTOR SYMPTOMS (VMS) WYETH CORP (US) 2008-01-09 EP claimed
EP-1879887-A2 NPY ANTAGONISTS, PREPARATION AND USE Cerep (FR) 2008-01-23 EP disclosed
WO-2006108965-A2 NPY ANTAGONISTS, PREPARATION AND USE CEREP (FR) 2006-10-19 WO disclosed