SCHEMBL4689730

SCHEMBL4689730

N[C@@H](CCN1CC2CN(C(=O)c3cnc4ccccc4c3)CC2C1)c1ccccc1

nearest known ligand 0.51

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
DPP4 P27487 3/20 0.51
CAPN1 P07384 1/20 0.45
MGAM O43451 1/20 0.43
KDM2B Q8NHM5 1/20 0.43
CCL5 P13501 7/20 0.42
CCR5 P51681 6/20 0.41
HDAC3 O15379 1/20 0.41
HDAC4 P56524 1/20 0.41
HDAC1 Q13547 1/20 0.41
HDAC7 Q8WUI4 1/20 0.41
HDAC2 Q92769 1/20 0.41
HDAC10 Q969S8 1/20 0.41
HDAC11 Q96DB2 1/20 0.41
HDAC8 Q9BY41 1/20 0.41
HDAC6 Q9UBN7 1/20 0.41
HDAC9 Q9UKV0 1/20 0.41
HDAC5 Q9UQL6 1/20 0.41
DPP8 Q6V1X1 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4694361 0.88 DPP4 (0.50) DPP4CAPN1CCL5CCR5HDAC3
SCHEMBL4691220 0.84 DPP4 (0.50) DPP4CCL5CCR5
SCHEMBL4694458 0.83 CCR5 (0.53) CCL5CCR5
SCHEMBL4696398 0.81 GRIN2B (0.48) DPP4MGAMKDM2BCCL5CCR5
SCHEMBL4695119 0.80 HDAC3 (0.42) DPP4CCL5CCR5HDAC3HDAC4
SCHEMBL3283162 0.79 CHRNB2 (0.54) CCL5CCR5
SCHEMBL5236953 0.79 DPP4 (0.50) DPP4CAPN1MGAMKDM2BHDAC3
SCHEMBL4693123 0.79 CCR5 (0.50) CCL5CCR5
SCHEMBL4694095 0.78 CCR5 (0.51) CCL5CCR5
SCHEMBL4695293 0.77 CCR5 (0.46) CCL5CCR5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1761542-B1 OCTAHYDROPYRROLO[3,4-C]PYRROLE DERIVATIVES AN THEIR USE AS ANTIVIRAL AGENTS HOFFMANN LA ROCHE (CH) 2008-01-02 EP claimed
EP-1761542-B1 OCTAHYDROPYRROLO[3,4-C]PYRROLE DERIVATIVES AN THEIR USE AS ANTIVIRAL AGENTS HOFFMANN LA ROCHE (CH) 2008-01-02 EP disclosed