SCHEMBL4696398

SCHEMBL4696398

N[C@@H](CCN1CC2CN(C(=O)c3ccc4ccccc4n3)CC2C1)c1ccccc1

nearest known ligand 0.48

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
GRIN2B Q13224 1/20 0.48
TSHR P16473 1/20 0.46
CCR5 P51681 6/20 0.42
MEN1 O00255 1/20 0.42
KMT2A Q03164 1/20 0.42
HCRTR1 O43613 1/20 0.42
HCRTR2 O43614 1/20 0.42
DPP4 P27487 1/20 0.42
DPP9 Q86TI2 1/20 0.42
MAPK1 P28482 1/20 0.42
RAB9A P51151 1/20 0.42
SMN1; SMN2 Q16637 1/20 0.42
ALDH1A1 P00352 1/20 0.42
GAA P10253 1/20 0.42
CCL5 P13501 5/20 0.41
KDM2B Q8NHM5 2/20 0.41
MGAM O43451 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4691220 0.86 DPP4 (0.50) CCR5HCRTR1HCRTR2DPP4CCL5
SCHEMBL4691767 0.81 CHRNB2 (0.54) CCR5CCL5
SCHEMBL4694458 0.81 CCR5 (0.53) CCR5CCL5
SCHEMBL4689730 0.81 DPP4 (0.51) CCR5DPP4CCL5KDM2BMGAM
SCHEMBL4690162 0.80 SMN1; SMN2 (0.49) CCR5SMN1; SMN2CCL5
SCHEMBL4694682 0.79 CCR5 (0.46) CCR5CCL5
SCHEMBL4695170 0.79 CYP2D6 (0.47) TSHRCCR5MEN1KMT2AMAPK1
SCHEMBL5237603 0.78 TSHR (0.46) GRIN2BTSHRMEN1KMT2AHCRTR1
SCHEMBL4691442 0.77 CCL5 (0.56) CCR5CCL5
SCHEMBL4694209 0.77 CCR5 (0.43) CCR5HCRTR1HCRTR2CCL5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1761542-B1 OCTAHYDROPYRROLO[3,4-C]PYRROLE DERIVATIVES AN THEIR USE AS ANTIVIRAL AGENTS HOFFMANN LA ROCHE (CH) 2008-01-02 EP claimed
EP-1761542-B1 OCTAHYDROPYRROLO[3,4-C]PYRROLE DERIVATIVES AN THEIR USE AS ANTIVIRAL AGENTS HOFFMANN LA ROCHE (CH) 2008-01-02 EP disclosed