SCHEMBL4690761

SCHEMBL4690761

NC(=O)c1nn(-c2ccccc2)nc1C(=O)N1CC2CN(CC[CH]c3ccccc3)C[C@H]2C1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 11/20 0.43
ALDH1A1 P00352 7/20 0.43
HPGD P15428 5/20 0.43
KMT2A Q03164 4/20 0.43
HSD17B10 Q99714 4/20 0.43
MEN1 O00255 3/20 0.43
ADORA2A P29274 4/20 0.42
LMNA P02545 1/20 0.42
ADORA3 P0DMS8 1/20 0.42
PKM P14618 1/20 0.42
ADORA2B P29275 1/20 0.42
ADORA1 P30542 1/20 0.42
KAT2B Q92831 1/20 0.42
HTT P42858 2/20 0.38
TSHR P16473 1/20 0.34
L3MBTL1 Q9Y468 1/20 0.34
CCR5 P51681 2/20 0.33
CCL5 P13501 1/20 0.33
MAPT P10636 1/20 0.33
MAOB P27338 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4694094 0.80 CHRNB2 (0.44) ALDH1A1HPGDL3MBTL1CCR5CHRNB2
SCHEMBL4694315 0.80 HCRTR2 (0.41) ALDH1A1KMT2A
SCHEMBL4694116 0.79 HCRTR2 (0.38) CCR5PARP1CHRNB2CHRNB4CHRNA3
SCHEMBL4691440 0.77 CCR5 (0.41) CCR5CCL5
SCHEMBL4690864 0.77 RIPK2 (0.40) HPGDKMT2AMEN1
SCHEMBL3282165 0.77 CCL5 (0.51) CCR5CCL5
SCHEMBL3290289 0.77 CCL5 (0.51) CCR5CCL5
SCHEMBL4690538 0.77 CCL5 (0.36) CCR5CCL5
SCHEMBL4693281 0.77 CHRNB2 (0.43) KMT2AHSD17B10MEN1LMNATSHR
SCHEMBL4692781 0.77 PKM (0.36) ALDH1A1HPGDKMT2AHSD17B10MEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1761542-B1 OCTAHYDROPYRROLO[3,4-C]PYRROLE DERIVATIVES AN THEIR USE AS ANTIVIRAL AGENTS HOFFMANN LA ROCHE (CH) 2008-01-02 EP claimed
EP-1761542-A2 OCTAHYDROPYRROLO[3,4-C]PYRROLE DERIVATIVES AN THEIR USE AS ANTIVIRAL AGENTS F.HOFFMANN-LA ROCHE AG (CH) 2007-03-14 EP claimed
WO-2005121145-A2 OCTAHYDRO-PYRROLO[3,4-C] DERIVATIVES AND THEIR USE AS ANTIVIRAL COMPOUNDS F. HOFFMANN-LA ROCHE AG (CH) 2005-12-22 WO claimed
EP-1761542-B1 OCTAHYDROPYRROLO[3,4-C]PYRROLE DERIVATIVES AN THEIR USE AS ANTIVIRAL AGENTS HOFFMANN LA ROCHE (CH) 2008-01-02 EP disclosed