SCHEMBL4690538

SCHEMBL4690538

Cn1nc(C(N)=O)cc1C(=O)N1CC2CN(CC[CH]c3ccccc3)C[C@H]2C1

nearest known ligand 0.36

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
CCL5 P13501 9/20 0.36
PLA2G10 O15496 2/20 0.36
HCRTR1 O43613 2/20 0.36
HCRTR2 O43614 2/20 0.36
CCR5 P51681 9/20 0.35
GSK3B P49841 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4692820 0.89 CCL5 (0.35) CCL5HCRTR1HCRTR2CCR5
SCHEMBL4690500 0.84 F10 (0.43)
SCHEMBL4690459 0.80 MEN1 (0.37) CCL5HCRTR1HCRTR2CCR5
SCHEMBL4694094 0.80 CHRNB2 (0.44) CCR5
SCHEMBL4694116 0.79 HCRTR2 (0.38) HCRTR1HCRTR2CCR5
SCHEMBL4693281 0.78 CHRNB2 (0.43) CCR5
SCHEMBL4693120 0.78 CCR5 (0.39) CCL5HCRTR1HCRTR2CCR5
SCHEMBL4690155 0.78 MEN1 (0.38) CCL5CCR5
SCHEMBL4696489 0.77 CCR5 (0.42) CCL5HCRTR1HCRTR2CCR5
SCHEMBL4693574 0.77 CCR5 (0.40) HCRTR1HCRTR2CCR5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1761542-B1 OCTAHYDROPYRROLO[3,4-C]PYRROLE DERIVATIVES AN THEIR USE AS ANTIVIRAL AGENTS HOFFMANN LA ROCHE (CH) 2008-01-02 EP disclosed