SCHEMBL4691302

SCHEMBL4691302

COc1c(C)cccc1C(=O)N1CC2CN(C(CC(N)=O)c3ccc(C)c(Cl)c3)CC2C1

nearest known ligand 0.42

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
HCRTR1 O43613 9/20 0.42
HCRTR2 O43614 9/20 0.42
CBX7 O95931 4/20 0.36
TNF P01375 2/20 0.36
GBA1 P04062 1/20 0.35
PDE4A P27815 1/20 0.35
PDE4B Q07343 1/20 0.35
PDE4C Q08493 1/20 0.35
PDE4D Q08499 1/20 0.35
NPC1 O15118 1/20 0.35
MAPT P10636 1/20 0.35
NFKB1 P19838 1/20 0.35
RAB9A P51151 1/20 0.35
NFKB2 Q00653 1/20 0.35
RELA Q04206 1/20 0.35
SMN1; SMN2 Q16637 1/20 0.35
CCR5 P51681 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4692627 0.94 HCRTR1 (0.50) HCRTR1HCRTR2CBX7NPC1RAB9A
SCHEMBL4693952 0.90 HCRTR1 (0.50) HCRTR1HCRTR2TNFPDE4APDE4B
SCHEMBL4691868 0.90 HCRTR1 (0.47) HCRTR1HCRTR2TNFGBA1MAPT
SCHEMBL4692886 0.90 ALDH1A1 (0.42) HCRTR1HCRTR2TNFGBA1MAPT
SCHEMBL4691405 0.89 HCRTR1 (0.48) HCRTR1HCRTR2TNFPDE4APDE4B
SCHEMBL4694354 0.88 P2RX7 (0.44) HCRTR1HCRTR2TNF
SCHEMBL3281863 0.87 HCRTR1 (0.48) HCRTR1HCRTR2TNFCCR5
SCHEMBL4693896 0.86 HCRTR1 (0.47) HCRTR1HCRTR2TNFPDE4APDE4B
SCHEMBL4693139 0.86 HCRTR1 (0.45) HCRTR1HCRTR2NPC1MAPT
SCHEMBL4695647 0.86 HCRTR1 (0.48) HCRTR1HCRTR2TNF

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1761542-B1 OCTAHYDROPYRROLO[3,4-C]PYRROLE DERIVATIVES AN THEIR USE AS ANTIVIRAL AGENTS HOFFMANN LA ROCHE (CH) 2008-01-02 EP claimed
EP-1761542-A2 OCTAHYDROPYRROLO[3,4-C]PYRROLE DERIVATIVES AN THEIR USE AS ANTIVIRAL AGENTS F.HOFFMANN-LA ROCHE AG (CH) 2007-03-14 EP claimed
WO-2005121145-A2 OCTAHYDRO-PYRROLO[3,4-C] DERIVATIVES AND THEIR USE AS ANTIVIRAL COMPOUNDS F. HOFFMANN-LA ROCHE AG (CH) 2005-12-22 WO claimed
EP-1761542-B1 OCTAHYDROPYRROLO[3,4-C]PYRROLE DERIVATIVES AN THEIR USE AS ANTIVIRAL AGENTS HOFFMANN LA ROCHE (CH) 2008-01-02 EP disclosed