SCHEMBL4691883

SCHEMBL4691883

Cc1ccc(NCCCN2CC3CN(C(=O)c4ccc(C(F)(F)F)c(F)c4)CC3C2)cc1Cl

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
BRAF P15056 3/20 0.41
RAF1 P04049 2/20 0.41
ARAF P10398 2/20 0.41
ALDH1A1 P00352 6/20 0.39
MAPT P10636 4/20 0.39
LMNA P02545 1/20 0.39
GAA P10253 1/20 0.39
HTT P42858 1/20 0.39
SMN1; SMN2 Q16637 1/20 0.39
UBE2M P61081 1/20 0.38
DCUN1D1 Q96GG9 1/20 0.38
AGTR1 P30556 1/20 0.37
EPHX2 P34913 2/20 0.37
HSD11B1 P28845 1/20 0.36
MEN1 O00255 1/20 0.36
POLB P06746 1/20 0.36
KMT2A Q03164 1/20 0.36
HPGD P15428 1/20 0.36
CNR2 P34972 2/20 0.36
GPR183 P32249 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4691230 0.93 UBE2M (0.40) BRAFRAF1ARAFALDH1A1MAPT
SCHEMBL4695365 0.88 BRAF (0.39) BRAFRAF1ARAFALDH1A1MAPT
SCHEMBL4690845 0.88 NPY2R (0.46) ALDH1A1MAPTLMNAGAAHTT
SCHEMBL4691875 0.87 CYP3A4 (0.46) ALDH1A1MAPTLMNAHTTUBE2M
SCHEMBL4693170 0.86 HCRTR1 (0.51) BRAFRAF1ARAFALDH1A1MAPT
SCHEMBL4694245 0.85 MAPT (0.43) BRAFRAF1ARAFALDH1A1MAPT
SCHEMBL4694155 0.85 NPY2R (0.48) ALDH1A1MAPTLMNAHTTSMN1; SMN2
SCHEMBL4691224 0.85 UBE2M (0.45) ALDH1A1MAPTLMNAGAAHTT
SCHEMBL4695756 0.84 RHOA (0.41) ALDH1A1MAPTLMNAGAAHTT
SCHEMBL4692110 0.84 HCRTR1 (0.51) BRAFRAF1ARAFALDH1A1MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1761542-B1 OCTAHYDROPYRROLO[3,4-C]PYRROLE DERIVATIVES AN THEIR USE AS ANTIVIRAL AGENTS HOFFMANN LA ROCHE (CH) 2008-01-02 EP claimed
EP-1761542-A2 OCTAHYDROPYRROLO[3,4-C]PYRROLE DERIVATIVES AN THEIR USE AS ANTIVIRAL AGENTS F.HOFFMANN-LA ROCHE AG (CH) 2007-03-14 EP claimed
WO-2005121145-A2 OCTAHYDRO-PYRROLO[3,4-C] DERIVATIVES AND THEIR USE AS ANTIVIRAL COMPOUNDS F. HOFFMANN-LA ROCHE AG (CH) 2005-12-22 WO claimed
EP-1761542-B1 OCTAHYDROPYRROLO[3,4-C]PYRROLE DERIVATIVES AN THEIR USE AS ANTIVIRAL AGENTS HOFFMANN LA ROCHE (CH) 2008-01-02 EP disclosed