SCHEMBL4694155

SCHEMBL4694155

Cc1ccc(NCCCN2CC3CN(C(=O)c4cccc(C(F)(F)F)c4)CC3C2)cc1Cl

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPY2R P49146 1/20 0.48
LCK P06239 1/20 0.46
MAPK14 Q16539 1/20 0.46
KCNK3 O14649 1/20 0.45
KCNK9 Q9NPC2 1/20 0.45
CHRM4 P08173 1/20 0.45
CHRM5 P08912 1/20 0.45
CHRM1 P11229 1/20 0.45
CHRM3 P20309 1/20 0.45
LMNA P02545 3/20 0.44
POLB P06746 2/20 0.44
SMN1; SMN2 Q16637 1/20 0.44
HPGD P15428 1/20 0.43
ALDH1A1 P00352 1/20 0.43
MAPT P10636 1/20 0.43
CCR2 P41597 3/20 0.43
MGLL Q99685 1/20 0.43
KMT2A Q03164 2/20 0.42
KDM4E B2RXH2 1/20 0.42
OPRM1 P35372 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4690845 0.90 NPY2R (0.46) NPY2RLMNASMN1; SMN2ALDH1A1MAPT
SCHEMBL4695756 0.89 RHOA (0.41) NPY2RLCKMAPK14CHRM4CHRM1
SCHEMBL4691640 0.88 MAPT (0.54) LMNASMN1; SMN2ALDH1A1MAPTKDM4E
SCHEMBL4694150 0.87 NPY2R (0.51) NPY2RKCNK3KCNK9CHRM4CHRM5
SCHEMBL4693613 0.87 GFER (0.49) NPY2RKCNK3KCNK9POLBSMN1; SMN2
SCHEMBL4695952 0.86 MAPT (0.43) LMNASMN1; SMN2ALDH1A1MAPTHTT
SCHEMBL4691883 0.85 BRAF (0.41) LMNAPOLBSMN1; SMN2HPGDALDH1A1
SCHEMBL4691230 0.85 UBE2M (0.40) LMNAPOLBSMN1; SMN2HPGDALDH1A1
SCHEMBL3281865 0.84 CCR5 (0.52) LMNASMN1; SMN2ALDH1A1MAPTHTT
SCHEMBL4694025 0.83 P2RX7 (0.48)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1761542-B1 OCTAHYDROPYRROLO[3,4-C]PYRROLE DERIVATIVES AN THEIR USE AS ANTIVIRAL AGENTS HOFFMANN LA ROCHE (CH) 2008-01-02 EP claimed
EP-1761542-A2 OCTAHYDROPYRROLO[3,4-C]PYRROLE DERIVATIVES AN THEIR USE AS ANTIVIRAL AGENTS F.HOFFMANN-LA ROCHE AG (CH) 2007-03-14 EP claimed
WO-2005121145-A2 OCTAHYDRO-PYRROLO[3,4-C] DERIVATIVES AND THEIR USE AS ANTIVIRAL COMPOUNDS F. HOFFMANN-LA ROCHE AG (CH) 2005-12-22 WO claimed
EP-1761542-B1 OCTAHYDROPYRROLO[3,4-C]PYRROLE DERIVATIVES AN THEIR USE AS ANTIVIRAL AGENTS HOFFMANN LA ROCHE (CH) 2008-01-02 EP disclosed