SCHEMBL4694658

SCHEMBL4694658

NC(=O)CNCc1ccc(CC(=O)NCCOC(=O)N(c2ccccc2-c2ccccc2)N2CC[CH]CC2)cc1

nearest known ligand 0.36

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 5/20 0.36
LMNA P02545 2/20 0.36
SPHK2 Q9NRA0 1/20 0.34
SPHK1 Q9NYA1 1/20 0.34
BACE1 P56817 1/20 0.33
THRB P10828 2/20 0.33
MEN1 O00255 1/20 0.33
KMT2A Q03164 1/20 0.33
PDCD1 Q15116 2/20 0.32
CD274 Q9NZQ7 2/20 0.32
MCL1 Q07820 2/20 0.32
TRPV1 Q8NER1 1/20 0.32
SCN3A Q9NY46 1/20 0.32
MAPT P10636 1/20 0.31
HPGD P15428 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4692679 0.91 PDCD1 (0.41) ALDH1A1LMNABACE1THRBMEN1
SCHEMBL6027362 0.87 TRPV1 (0.39) ALDH1A1LMNAPDCD1CD274TRPV1
SCHEMBL4695551 0.83 CNR2 (0.40) LMNAMEN1KMT2APDCD1CD274
SCHEMBL6027475 0.82 TRPV1 (0.37) LMNATRPV1HPGD
SCHEMBL4691773 0.81 KDM4E (0.41) ALDH1A1LMNAMEN1KMT2APDCD1
SCHEMBL4695176 0.81 POLB (0.37) ALDH1A1LMNAKMT2AHPGD
SCHEMBL4696335 0.78 PDCD1 (0.44) ALDH1A1PDCD1CD274
SCHEMBL5805321 0.78 HDAC3 (0.40) TRPV1
SCHEMBL5722183 0.78 HPGD (0.40) ALDH1A1LMNASPHK2SPHK1MEN1
SCHEMBL6027738 0.77 ESRRG (0.40) PDCD1CD274MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1893577-A1 BIPHENYL COMPOUNDS USEFUL AS MUSCARINIC RECEPTOR ANTAGONISTS Theravance, Inc. (US) 2008-03-05 EP claimed
WO-2006138218-A1 BIPHENYL COMPOUNDS USEFUL AS MUSCARINIC RECEPTOR ANTAGONISTS THERAVANCE, INC. (US) 2006-12-28 WO claimed