SCHEMBL4692108

SCHEMBL4692108

Cc1ccc(C(CC(N)=O)N2CC3CN(C(=O)c4c(C)nc(-c5ccccc5)nc4C)CC3C2)cc1Cl

nearest known ligand 0.40

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
HCRTR1 O43613 4/20 0.40
HCRTR2 O43614 4/20 0.40
CCR5 P51681 9/20 0.38
CHRM2 P08172 1/20 0.38
CCL5 P13501 9/20 0.37
TNF P01375 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4696341 0.92 HCRTR1 (0.37) HCRTR1HCRTR2CCR5CHRM2CCL5
SCHEMBL3283594 0.86 CCL5 (0.43) CCR5CCL5
SCHEMBL3281863 0.85 HCRTR1 (0.48) HCRTR1HCRTR2CCR5TNF
SCHEMBL4689556 0.84 LMNA (0.50) HCRTR1HCRTR2
SCHEMBL4695130 0.83 KMT2A (0.43) HCRTR1HCRTR2CCR5
SCHEMBL4693079 0.83 HCRTR1 (0.38) HCRTR1HCRTR2CCR5CCL5TNF
SCHEMBL4694334 0.83 HCRTR1 (0.43) HCRTR1HCRTR2CCR5CCL5TNF
SCHEMBL4690403 0.83 HCRTR1 (0.39) HCRTR1HCRTR2CCR5TNF
SCHEMBL3282223 0.82 CCR5 (0.43) HCRTR1HCRTR2CCR5CHRM2CCL5
SCHEMBL4694788 0.82 HCRTR1 (0.45) HCRTR1HCRTR2CCR5TNF

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1761542-B1 OCTAHYDROPYRROLO[3,4-C]PYRROLE DERIVATIVES AN THEIR USE AS ANTIVIRAL AGENTS HOFFMANN LA ROCHE (CH) 2008-01-02 EP claimed
EP-1761542-B1 OCTAHYDROPYRROLO[3,4-C]PYRROLE DERIVATIVES AN THEIR USE AS ANTIVIRAL AGENTS HOFFMANN LA ROCHE (CH) 2008-01-02 EP disclosed