SCHEMBL4696341

SCHEMBL4696341

Cc1ccc(C(CC(N)=O)N2CC3CN(C(=O)c4c(C)nc(-c5ccncc5)nc4C)CC3C2)cc1Cl

nearest known ligand 0.37

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
HCRTR1 O43613 8/20 0.37
HCRTR2 O43614 8/20 0.37
CCR5 P51681 5/20 0.37
NPC1 O15118 1/20 0.34
RAB9A P51151 1/20 0.34
DPP4 P27487 2/20 0.34
CHRM2 P08172 1/20 0.33
PDE4B Q07343 1/20 0.33
TNF P01375 1/20 0.32
KCNH2 Q12809 1/20 0.32
CCL5 P13501 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4692108 0.92 HCRTR1 (0.40) HCRTR1HCRTR2CCR5CHRM2TNF
SCHEMBL4695972 0.89 CHRNB2 (0.40) HCRTR1HCRTR2NPC1TNF
SCHEMBL3283594 0.85 CCL5 (0.43) CCR5KCNH2CCL5
SCHEMBL3282223 0.84 CCR5 (0.43) HCRTR1HCRTR2CCR5CHRM2CCL5
SCHEMBL4693079 0.82 HCRTR1 (0.38) HCRTR1HCRTR2CCR5PDE4BTNF
SCHEMBL3281863 0.82 HCRTR1 (0.48) HCRTR1HCRTR2CCR5TNFKCNH2
SCHEMBL4690403 0.82 HCRTR1 (0.39) HCRTR1HCRTR2CCR5PDE4BTNF
SCHEMBL4694334 0.82 HCRTR1 (0.43) HCRTR1HCRTR2CCR5TNFCCL5
SCHEMBL4693625 0.82 HCRTR1 (0.37) HCRTR1HCRTR2DPP4TNF
SCHEMBL4691396 0.82 HCRTR1 (0.39) HCRTR1HCRTR2DPP4TNF

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1761542-B1 OCTAHYDROPYRROLO[3,4-C]PYRROLE DERIVATIVES AN THEIR USE AS ANTIVIRAL AGENTS HOFFMANN LA ROCHE (CH) 2008-01-02 EP claimed
EP-1761542-B1 OCTAHYDROPYRROLO[3,4-C]PYRROLE DERIVATIVES AN THEIR USE AS ANTIVIRAL AGENTS HOFFMANN LA ROCHE (CH) 2008-01-02 EP disclosed