SCHEMBL4692182

SCHEMBL4692182

NC(=O)C1[C@@H]2CN(C(=O)c3cccc4cccnc34)CC2CN1CC[CH]c1ccccc1

nearest known ligand 0.47

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
HCRTR1 O43613 12/20 0.47
HCRTR2 O43614 10/20 0.47
PARP1 P09874 1/20 0.38
HTR2A P28223 1/20 0.36
HTR2C P28335 1/20 0.36
PKLR P30613 1/20 0.35
ALDH1A1 P00352 2/20 0.35
CCR3 P51677 1/20 0.34
KDM4E B2RXH2 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5236228 0.88 HCRTR2 (0.45) HCRTR1HCRTR2ALDH1A1
SCHEMBL4691766 0.84 CHRNB2 (0.47) ALDH1A1KDM4E
SCHEMBL4694358 0.83 DPP4 (0.45) HTR2AALDH1A1CCR3
SCHEMBL5231921 0.83 P2RX7 (0.40) ALDH1A1KDM4E
SCHEMBL5232784 0.82 CHRNB2 (0.43) ALDH1A1
SCHEMBL4693442 0.82 EIF4A3 (0.37) HCRTR1HCRTR2CCR3
SCHEMBL3283159 0.80 CHRNB2 (0.47) ALDH1A1KDM4E
SCHEMBL4691769 0.80 CYP2C9 (0.41) HCRTR1HCRTR2
SCHEMBL4696396 0.80 TSHR (0.41) HCRTR1HCRTR2ALDH1A1KDM4E
SCHEMBL4695167 0.80 CYP2D6 (0.38) ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1761542-B1 OCTAHYDROPYRROLO[3,4-C]PYRROLE DERIVATIVES AN THEIR USE AS ANTIVIRAL AGENTS HOFFMANN LA ROCHE (CH) 2008-01-02 EP claimed
EP-1761542-A2 OCTAHYDROPYRROLO[3,4-C]PYRROLE DERIVATIVES AN THEIR USE AS ANTIVIRAL AGENTS F.HOFFMANN-LA ROCHE AG (CH) 2007-03-14 EP claimed
WO-2005121145-A2 OCTAHYDRO-PYRROLO[3,4-C] DERIVATIVES AND THEIR USE AS ANTIVIRAL COMPOUNDS F. HOFFMANN-LA ROCHE AG (CH) 2005-12-22 WO claimed
EP-1761542-B1 OCTAHYDROPYRROLO[3,4-C]PYRROLE DERIVATIVES AN THEIR USE AS ANTIVIRAL AGENTS HOFFMANN LA ROCHE (CH) 2008-01-02 EP disclosed