SCHEMBL4696396

SCHEMBL4696396

NC(=O)C1[C@@H]2CN(C(=O)c3ccc4ccccc4n3)CC2CN1CC[CH]c1ccccc1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TSHR P16473 1/20 0.41
GRIN2B Q13224 1/20 0.39
ALDH1A1 P00352 3/20 0.37
GAA P10253 3/20 0.37
MGAM O43451 1/20 0.37
MAPK1 P28482 1/20 0.37
RAB9A P51151 1/20 0.37
SMN1; SMN2 Q16637 1/20 0.37
MEN1 O00255 2/20 0.36
KMT2A Q03164 2/20 0.36
HCRTR1 O43613 1/20 0.36
HCRTR2 O43614 1/20 0.36
MAPT P10636 2/20 0.35
KDM4E B2RXH2 1/20 0.35
HPGD P15428 1/20 0.35
TPSAB1 Q15661 1/20 0.35
TPSD1 Q9BZJ3 1/20 0.35
TPSG1 Q9NRR2 1/20 0.35
L3MBTL1 Q9Y468 1/20 0.35
KDM2B Q8NHM5 2/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4691215 0.88 DPP4 (0.44) ALDH1A1HCRTR1HCRTR2HPGDDPP4
SCHEMBL5232784 0.84 CHRNB2 (0.43) ALDH1A1SMN1; SMN2MEN1KMT2AHPGD
SCHEMBL4691766 0.84 CHRNB2 (0.47) ALDH1A1GAARAB9ASMN1; SMN2MAPT
SCHEMBL4689727 0.83 DPP4 (0.45) MGAMRAB9AKDM2BDPP4
SCHEMBL4695167 0.82 CYP2D6 (0.38) ALDH1A1GAA
SCHEMBL4693442 0.80 EIF4A3 (0.37) HCRTR1HCRTR2MAPT
SCHEMBL4694358 0.80 DPP4 (0.45) ALDH1A1SMN1; SMN2HPGDDPP4
SCHEMBL5235592 0.80 RAB9A (0.47) GRIN2BALDH1A1GAARAB9ASMN1; SMN2
SCHEMBL4692182 0.80 HCRTR1 (0.47) ALDH1A1HCRTR1HCRTR2KDM4E
SCHEMBL5231921 0.79 P2RX7 (0.40) ALDH1A1GAARAB9AMEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1761542-B1 OCTAHYDROPYRROLO[3,4-C]PYRROLE DERIVATIVES AN THEIR USE AS ANTIVIRAL AGENTS HOFFMANN LA ROCHE (CH) 2008-01-02 EP claimed
EP-1761542-A2 OCTAHYDROPYRROLO[3,4-C]PYRROLE DERIVATIVES AN THEIR USE AS ANTIVIRAL AGENTS F.HOFFMANN-LA ROCHE AG (CH) 2007-03-14 EP claimed
WO-2005121145-A2 OCTAHYDRO-PYRROLO[3,4-C] DERIVATIVES AND THEIR USE AS ANTIVIRAL COMPOUNDS F. HOFFMANN-LA ROCHE AG (CH) 2005-12-22 WO claimed