SCHEMBL4692334

SCHEMBL4692334

CCOc1ccccc1C(=O)N1CC2CN(C(CC(N)=O)c3ccc(C)c(Cl)c3)CC2C1

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HCRTR1 O43613 7/20 0.51
HCRTR2 O43614 7/20 0.51
NPSR1 Q6W5P4 3/20 0.46
NOD2 Q9HC29 1/20 0.46
LMNA P02545 2/20 0.44
SMN1; SMN2 Q16637 2/20 0.44
TSHR P16473 2/20 0.44
RAB9A P51151 1/20 0.44
TNF P01375 1/20 0.42
PDE4A P27815 1/20 0.41
PDE4B Q07343 1/20 0.41
PDE4C Q08493 1/20 0.41
PDE4D Q08499 1/20 0.41
CHRM2 P08172 1/20 0.40
CHRM3 P20309 1/20 0.40
HTT P42858 1/20 0.40
TDP1 Q9NUW8 1/20 0.40
ALOX15 P16050 1/20 0.39
HSD17B10 Q99714 1/20 0.39
MEN1 O00255 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4691405 0.91 HCRTR1 (0.48) HCRTR1HCRTR2TSHRTNFPDE4A
SCHEMBL4692886 0.88 ALDH1A1 (0.42) HCRTR1HCRTR2NPSR1TNFHTT
SCHEMBL4693693 0.88 HCRTR1 (0.51) HCRTR1HCRTR2TNF
SCHEMBL4693484 0.88 HCRTR1 (0.48) HCRTR1HCRTR2TNFMEN1KMT2A
SCHEMBL4693952 0.87 HCRTR1 (0.50) HCRTR1HCRTR2TSHRTNFPDE4A
SCHEMBL4691904 0.86 HCRTR1 (0.46) HCRTR1HCRTR2LMNATSHRTNF
SCHEMBL4694224 0.86 TNF (0.39) HCRTR1HCRTR2NPSR1TNF
SCHEMBL4692627 0.85 HCRTR1 (0.50) HCRTR1HCRTR2NPSR1LMNASMN1; SMN2
SCHEMBL4691868 0.85 HCRTR1 (0.47) HCRTR1HCRTR2LMNASMN1; SMN2TNF
SCHEMBL4694354 0.85 P2RX7 (0.44) HCRTR1HCRTR2TNF

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1761542-B1 OCTAHYDROPYRROLO[3,4-C]PYRROLE DERIVATIVES AN THEIR USE AS ANTIVIRAL AGENTS HOFFMANN LA ROCHE (CH) 2008-01-02 EP claimed
EP-1761542-B1 OCTAHYDROPYRROLO[3,4-C]PYRROLE DERIVATIVES AN THEIR USE AS ANTIVIRAL AGENTS HOFFMANN LA ROCHE (CH) 2008-01-02 EP disclosed
EP-1761542-A2 OCTAHYDROPYRROLO[3,4-C]PYRROLE DERIVATIVES AN THEIR USE AS ANTIVIRAL AGENTS F.HOFFMANN-LA ROCHE AG (CH) 2007-03-14 EP disclosed
WO-2005121145-A2 OCTAHYDRO-PYRROLO[3,4-C] DERIVATIVES AND THEIR USE AS ANTIVIRAL COMPOUNDS F. HOFFMANN-LA ROCHE AG (CH) 2005-12-22 WO disclosed