SCHEMBL4692853

SCHEMBL4692853

Cc1ccc(NCCCN2CC3CN(C(=O)c4cc5ccccc5o4)CC3C2)cc1Cl

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
RAB9A P51151 3/20 0.52
L3MBTL1 Q9Y468 3/20 0.52
NPC1 O15118 2/20 0.52
HRH4 Q9H3N8 1/20 0.46
ALDH1A1 P00352 5/20 0.45
NPSR1 Q6W5P4 4/20 0.45
MEN1 O00255 2/20 0.45
KMT2A Q03164 2/20 0.45
GLA P06280 1/20 0.45
GAA P10253 1/20 0.45
HPGD P15428 4/20 0.45
SMN1; SMN2 Q16637 4/20 0.45
MAPT P10636 4/20 0.43
POLB P06746 1/20 0.43
USP2 O75604 3/20 0.43
KDM4E B2RXH2 3/20 0.43
LMNA P02545 3/20 0.43
TP53 P04637 3/20 0.43
MAPK1 P28482 3/20 0.43
HTT P42858 3/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4692849 0.86 DRD3 (0.49) RAB9AL3MBTL1NPC1SLC6A2SLC6A4
SCHEMBL4691763 0.84 KMT2A (0.56) RAB9ANPC1ALDH1A1NPSR1MEN1
SCHEMBL4695249 0.84 RECQL (0.48) RAB9AL3MBTL1NPC1ALDH1A1MEN1
SCHEMBL4691640 0.84 MAPT (0.54) RAB9AALDH1A1NPSR1GAASMN1; SMN2
SCHEMBL4692889 0.83 MAPT (0.45) ALDH1A1GAAHPGDSMN1; SMN2MAPT
SCHEMBL4693334 0.83 ALDH1A1 (0.45) ALDH1A1KMT2AGAASMN1; SMN2MAPT
SCHEMBL4692171 0.82 HDAC6 (0.41) L3MBTL1ALDH1A1MEN1KMT2AGAA
SCHEMBL3281865 0.82 CCR5 (0.52) ALDH1A1GAASMN1; SMN2MAPTLMNA
SCHEMBL4690668 0.81 ALDH1A1 (0.43) RAB9AL3MBTL1NPC1ALDH1A1MEN1
SCHEMBL4691905 0.81 HCRTR1 (0.47) RAB9ANPC1ALDH1A1MEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1761542-B1 OCTAHYDROPYRROLO[3,4-C]PYRROLE DERIVATIVES AN THEIR USE AS ANTIVIRAL AGENTS HOFFMANN LA ROCHE (CH) 2008-01-02 EP claimed
EP-1761542-A2 OCTAHYDROPYRROLO[3,4-C]PYRROLE DERIVATIVES AN THEIR USE AS ANTIVIRAL AGENTS F.HOFFMANN-LA ROCHE AG (CH) 2007-03-14 EP claimed
WO-2005121145-A2 OCTAHYDRO-PYRROLO[3,4-C] DERIVATIVES AND THEIR USE AS ANTIVIRAL COMPOUNDS F. HOFFMANN-LA ROCHE AG (CH) 2005-12-22 WO claimed
EP-1761542-B1 OCTAHYDROPYRROLO[3,4-C]PYRROLE DERIVATIVES AN THEIR USE AS ANTIVIRAL AGENTS HOFFMANN LA ROCHE (CH) 2008-01-02 EP disclosed