SCHEMBL4691763

SCHEMBL4691763

Cc1ccc(NCCCN2CC3CN(C(=O)c4ccco4)CC3C2)cc1Cl

nearest known ligand 0.56

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 5/20 0.56
ALDH1A1 P00352 5/20 0.49
USP2 O75604 2/20 0.49
MAPT P10636 2/20 0.49
NPSR1 Q6W5P4 2/20 0.49
MEN1 O00255 1/20 0.46
CHRNB2 P17787 1/20 0.43
CHRNB4 P30926 1/20 0.43
CHRNA3 P32297 1/20 0.43
CHRNA7 P36544 1/20 0.43
CHRNA4 P43681 1/20 0.43
LMNA P02545 2/20 0.43
TSHR P16473 1/20 0.43
NPC1 O15118 2/20 0.43
RAB9A P51151 2/20 0.43
ATM Q13315 1/20 0.43
SMN1; SMN2 Q16637 2/20 0.42
HTT P42858 1/20 0.42
GAA P10253 1/20 0.42
POLB P06746 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4692728 0.86 CHRNB2 (0.47) KMT2AALDH1A1MAPTCHRNB2CHRNB4
SCHEMBL4691755 0.85 KMT2A (0.62) KMT2AALDH1A1USP2MAPTNPSR1
SCHEMBL4691640 0.85 MAPT (0.54) ALDH1A1MAPTNPSR1LMNARAB9A
SCHEMBL3281865 0.85 CCR5 (0.52) ALDH1A1MAPTLMNASMN1; SMN2HTT
SCHEMBL4692853 0.84 RAB9A (0.52) KMT2AALDH1A1USP2MAPTNPSR1
SCHEMBL4693334 0.84 ALDH1A1 (0.45) KMT2AALDH1A1MAPTLMNASMN1; SMN2
SCHEMBL4692889 0.84 MAPT (0.45) ALDH1A1USP2MAPTLMNASMN1; SMN2
SCHEMBL4691642 0.83 CCR5 (0.47) KMT2AALDH1A1MAPTCHRNB2CHRNB4
SCHEMBL14436612 0.83 ALDH1A1 (0.45) KMT2AALDH1A1MAPTMEN1LMNA
SCHEMBL4691511 0.83 CCR5 (0.54) ALDH1A1MAPTLMNAGAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1761542-B1 OCTAHYDROPYRROLO[3,4-C]PYRROLE DERIVATIVES AN THEIR USE AS ANTIVIRAL AGENTS HOFFMANN LA ROCHE (CH) 2008-01-02 EP claimed
EP-1761542-A2 OCTAHYDROPYRROLO[3,4-C]PYRROLE DERIVATIVES AN THEIR USE AS ANTIVIRAL AGENTS F.HOFFMANN-LA ROCHE AG (CH) 2007-03-14 EP claimed
WO-2005121145-A2 OCTAHYDRO-PYRROLO[3,4-C] DERIVATIVES AND THEIR USE AS ANTIVIRAL COMPOUNDS F. HOFFMANN-LA ROCHE AG (CH) 2005-12-22 WO claimed
EP-1761542-B1 OCTAHYDROPYRROLO[3,4-C]PYRROLE DERIVATIVES AN THEIR USE AS ANTIVIRAL AGENTS HOFFMANN LA ROCHE (CH) 2008-01-02 EP disclosed