SCHEMBL4693224

SCHEMBL4693224

CCCCCc1cc(C(F)(F)F)nnc1NC(=O)C(C)(C)C

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
S1PR1 P21453 2/20 0.43
LMNA P02545 1/20 0.35
SOAT1 P35610 2/20 0.33
PLK1 P53350 1/20 0.33
ALDH1A1 P00352 1/20 0.33
L3MBTL1 Q9Y468 1/20 0.33
CYP1A2 P05177 1/20 0.33
POLB P06746 1/20 0.33
CYP2C9 P11712 1/20 0.33
KDM4E B2RXH2 1/20 0.32
TP53 P04637 1/20 0.32
CYP3A4 P08684 1/20 0.32
MAPT P10636 1/20 0.32
ALOX15 P16050 1/20 0.32
TSHR P16473 1/20 0.32
ACAT1 P24752 1/20 0.32
FAAH O00519 1/20 0.32
CNR1 P21554 1/20 0.32
CNR2 P34972 1/20 0.32
ALPL P05186 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4694453 0.83 S1PR1 (0.38) S1PR1SOAT1ALDH1A1L3MBTL1CYP2C9
SCHEMBL4691170 0.80 AR (0.40) S1PR1SOAT1ALDH1A1KDM4ETP53
SCHEMBL3963194 0.74 L3MBTL1 (0.38) LMNAALDH1A1L3MBTL1CYP1A2POLB
SCHEMBL3966666 0.73 L3MBTL1 (0.36) LMNASOAT1ALDH1A1L3MBTL1KDM4E
SCHEMBL4689066 0.71 TLR8 (0.44)
SCHEMBL3967355 0.68 L3MBTL1 (0.39) LMNAALDH1A1L3MBTL1KDM4EMAPT
SCHEMBL8325829 0.67 CNR2 (0.47) SOAT1L3MBTL1MAPTCNR1CNR2
SCHEMBL28481299 0.65 PTGS2 (0.37) TP53CYP3A4MAPTALOX15TSHR
SCHEMBL21120072 0.64 GLS (0.50)
SCHEMBL4689750 0.63 SMN1; SMN2 (0.45) LMNAALDH1A1L3MBTL1CYP1A2POLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1879896-A1 IMIDAZOPYRIDAZINE COMPOUNDS ELI LILLY AND COMPANY (US) 2008-01-23 EP disclosed
WO-2006107784-A1 IMIDAZOPYRIDAZINE COMPOUNDS ELI LILLY AND COMPANY (US) 2006-10-12 WO disclosed